Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-methyltrienolone from androgen receptor (unknown origin) expressed in HEK293 cell lysate incubated overnight by microbeta scinti...More data for this Ligand-Target Pair
Affinity DataIC50: 0.302nMAssay Description:Agonist activity at GAL4 DNA-binding domain fused androgen receptor (unknown origin) ligand binding domain expressed in UAS-bla GripTite 293 cells as...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 3.09nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.680nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 288 KMore data for this Ligand-Target Pair
Affinity DataKd: 1.21nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 303 KMore data for this Ligand-Target Pair
Affinity DataKd: 0.610nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 273 KMore data for this Ligand-Target Pair
Affinity DataKd: 0.560nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 283 KMore data for this Ligand-Target Pair
Affinity DataKd: 1.95nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 310KMore data for this Ligand-Target Pair
Affinity DataKd: 0.740nMAssay Description:Dissociation constant value of the radiolabeled compound against the androgen receptor 293 KMore data for this Ligand-Target Pair
Affinity DataKd: 0.990nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 298 KMore data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Binding affinity to androgen receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.520nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 278 KMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0130nMAssay Description:Agonist activity at human androgen receptor expressed in mouse C2C12 cells cotransfected with GRE/ARE reporter plasmid assessed as receptor transacti...More data for this Ligand-Target Pair
Affinity DataKd: 1.51nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 308 KMore data for this Ligand-Target Pair