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Found 3 of affinity data with PDB=3G42
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(CHEMBL527018 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  140nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279255(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-methyl...)
Affinity DataIC50:  280nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Mus musculus (Mouse))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(CHEMBL527018 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of TACE in mouse Raw264.7 cells assessed as inhibition of LPS-induced TNFalpha production treated 1 hr before LPS challenge measured 4 hrs...More data for this Ligand-Target Pair