Affinity DataKi: 100nM ΔG°: -40.6kJ/moleT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at 30 °C with substrate, and test compounds in the presence of 100 uM ATP/ [gamma-32P...More data for this Ligand-Target Pair
Affinity DataKon: 0.0562M-1s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
Affinity DataKoff: 6.02E+5s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
Affinity DataKon: 0.0170M-1s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
Affinity DataKoff: 8.59E+4s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
Affinity DataKd: 3.97E+4nMpH: 7.5 T: 2°CAssay Description:ThermofluorMore data for this Ligand-Target Pair