Compile Data Set for Download or QSAR
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Found 788
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  16nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human Adk using [U-14C]adenosine by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of purified human adenosine kinase using varying levels of [3H]Ado as substrate in presence of adenosine deaminase inhibitor deoxycoformyc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of adhenosine kinaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368712(CHEMBL608051)
Affinity DataKi:  40nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368710(CHEMBL607761)
Affinity DataKi:  150nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368709(CHEMBL607766)
Affinity DataKi:  160nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368707(CHEMBL612205)
Affinity DataKi:  170nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533828(CHEMBL4570031)
Affinity DataKi:  184nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368708(CHEMBL611890)
Affinity DataKi:  300nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524383(CHEMBL4442160)
Affinity DataKi:  410nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524385(CHEMBL4463459)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50100587((2R,3R,4S,5R)-2-(6-Amino-5-nitro-pyrimidin-4-ylami...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of adenosine kinase from undialyzed W1-L2 lysate (0-50 uM)Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533823(CHEMBL494210)
Affinity DataKi:  5.04E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524391(CHEMBL2042164)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533825(CHEMBL4460819)
Affinity DataKi:  5.44E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533832(CHEMBL4524434)
Affinity DataKi:  5.64E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50368706(CHEMBL607762)
Affinity DataKi:  8.50E+3nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533830(CHEMBL4460655)
Affinity DataKi:  8.56E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533829(CHEMBL4592393)
Affinity DataKi:  8.75E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533827(CHEMBL4457103)
Affinity DataKi:  9.18E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533833(CHEMBL4545415)
Affinity DataKi:  1.11E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533831(CHEMBL4445820)
Affinity DataKi:  1.51E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533834(CHEMBL4448716)
Affinity DataKi:  1.95E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533824(CHEMBL4574016)
Affinity DataKi:  2.52E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533826(CHEMBL4520524)
Affinity DataKi:  2.54E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524392(CHEMBL4475059)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524386(CHEMBL4474951)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524384(CHEMBL4458246)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50456504(CHEMBL4214720)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524389(CHEMBL4525944)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524393(CHEMBL4448092)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524387(CHEMBL4566815)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524390(CHEMBL4475619)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50524388(CHEMBL4449169)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533474(CHEMBL4460859)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of human adenosine kinase assessed as reduction in conversion of adenosine to AMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human adenosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50:  0.100nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50178014(CHEMBL370164 | N-(4-chlorophenyl)-2-(5-phenyl-7-(5...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090843((1R,5S)-2-((3R,4aR)-4-Amino-5-bromo-pyrrolo[2,3-d]...)
Affinity DataIC50:  0.200nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090843((1R,5S)-2-((3R,4aR)-4-Amino-5-bromo-pyrrolo[2,3-d]...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090843((1R,5S)-2-((3R,4aR)-4-Amino-5-bromo-pyrrolo[2,3-d]...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human adenosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50174602((4R,5R,6S)-5-[4-(4-Fluoro-phenylamino)-5-phenyl-py...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50201834(5-benzo[b]thiophen-2-yl-6-(6-morpholin-4-ylpyridin...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50134740((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]-AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50134740((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50090887((1R,4S,5R)-2-Methyl-5-(5-phenyl-4-phenylamino-pyrr...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human adenosine kinase assessed as reduction in conversion of adenosine to AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50178003(CHEMBL370011 | N-cyclopropyl-2-(5-phenyl-7-(5-deox...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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