Compile Data Set for Download or QSAR
maximum 50k data
Found 119 of ec50 data for polymerid = 1024,50000929
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014777(1-Di-p-tolylmethyl-1H-imidazole | CHEMBL135381)
Affinity DataEC50:  6.40nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014754(1-[(4-Chloro-phenyl)-(4-methoxy-phenyl)-methyl]-1H...)
Affinity DataEC50:  8.40nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014780(1-[Bis-(4-chloro-phenyl)-methyl]-1H-[1,2,4]triazol...)
Affinity DataEC50:  8.80nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014773(1-[Bis-(4-bromo-phenyl)-methyl]-1H-imidazole | CHE...)
Affinity DataEC50:  8.90nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014803(4-[Bis-(4-chloro-phenyl)-methyl]-4H-[1,2,4]triazol...)
Affinity DataEC50:  9.30nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014776(1-[bis(4-chlorophenyl)(1H-imidazol-2-yl)methyl]-1H...)
Affinity DataEC50:  9.40nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014771(Bis-(4-chloro-phenyl)-thiazol-5-yl-methanol | CHEM...)
Affinity DataEC50:  9.60nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014764(5-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-1H-...)
Affinity DataEC50:  11nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014809(1-[(4-Chloro-phenyl)-(4-trifluoromethyl-phenyl)-me...)
Affinity DataEC50:  11nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014796(1-[(4-Methoxy-phenyl)-p-tolyl-methyl]-1H-imidazole...)
Affinity DataEC50:  11nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014763(4-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-1H-...)
Affinity DataEC50:  11nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014755(1-[Bis-(4-methoxy-phenyl)-methyl]-1H-imidazole | C...)
Affinity DataEC50:  13nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014800(1-[bis(4-chlorophenyl)(1H-imidazol-4-yl)methyl]-1H...)
Affinity DataEC50:  16nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014759(5-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-thi...)
Affinity DataEC50:  17nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014814(4-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-1H-...)
Affinity DataEC50:  18nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014804(Bis-(4-chloro-phenyl)-isothiazol-5-yl-methanol | C...)
Affinity DataEC50:  19nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014782(1-[Bis-(4-chloro-phenyl)-methyl]-1H-[1,2,3]triazol...)
Affinity DataEC50:  19nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014808(1-[(4-Chloro-phenyl)-phenyl-methyl]-1H-imidazole |...)
Affinity DataEC50:  20nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014775(5-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-pyr...)
Affinity DataEC50:  26nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014785(Bis-(4-chloro-phenyl)-(1H-imidazol-4-yl)-methanol ...)
Affinity DataEC50:  28nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014783(2-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-pyr...)
Affinity DataEC50:  29nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014778(Bis-(4-chloro-phenyl)-(1H-pyrazol-4-yl)-methanol |...)
Affinity DataEC50:  30nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014810(1-[Bis-(4-nitro-phenyl)-methyl]-1H-imidazole | CHE...)
Affinity DataEC50:  40nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014797(1-[Bis-(4-fluoro-phenyl)-methyl]-1H-imidazole | CH...)
Affinity DataEC50:  40nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014756(1-[Bis-(4-chloro-phenyl)-methyl]-1H-imidazole | CH...)
Affinity DataEC50:  42nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50367548(CHEMBL1794921)
Affinity DataEC50:  50nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014750(3-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-pyr...)
Affinity DataEC50:  50nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014802(4-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-pyr...)
Affinity DataEC50:  50nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014324(5-[Bis-(4-chloro-phenyl)-methyl]-pyrimidine | 5-[B...)
Affinity DataEC50:  55nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014324(5-[Bis-(4-chloro-phenyl)-methyl]-pyrimidine | 5-[B...)
Affinity DataEC50:  55nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014793(5-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-iso...)
Affinity DataEC50:  57nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014749(3-[Bis-(4-chloro-phenyl)-imidazol-1-yl-methyl]-1H-...)
Affinity DataEC50:  61nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014781(1-[(2-Methoxy-phenyl)-phenyl-methyl]-1H-imidazole ...)
Affinity DataEC50:  66nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50024481((4-Chloro-phenyl)-pyrimidin-5-yl-(4-trifluoromethy...)
Affinity DataEC50:  66nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014815(Bis-(4-chloro-phenyl)-pyrimidin-5-yl-methanol | CH...)
Affinity DataEC50:  71nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014815(Bis-(4-chloro-phenyl)-pyrimidin-5-yl-methanol | CH...)
Affinity DataEC50:  71nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014752(1-[Bis-(2-chloro-phenyl)-methyl]-1H-imidazole | CH...)
Affinity DataEC50:  76nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50024516(5-[Bis-(4-chloro-phenyl)-fluoro-methyl]-pyrimidine...)
Affinity DataEC50:  78nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50024524(5-[1,1-Bis-(4-chloro-phenyl)-ethyl]-pyrimidine | C...)
Affinity DataEC50:  82nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014794(3-[Bis-(4-chloro-phenyl)-methyl]-pyridine | CHEMBL...)
Affinity DataEC50:  84nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014798(Bis-(4-chloro-phenyl)-pyridin-4-yl-methanol | CHEM...)
Affinity DataEC50:  84nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014791(Bis-(4-chloro-phenyl)-(1H-pyrazol-3-yl)-methanol |...)
Affinity DataEC50:  90nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014774(Bis-(4-chloro-phenyl)-pyrazin-2-yl-methanol | CHEM...)
Affinity DataEC50:  94nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014788(1-Benzhydryl-1H-imidazole | CHEMBL336638)
Affinity DataEC50:  125nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50024513(6-Acetylsulfanyl-8-[2-[(4-amino-2-methyl-pyrimidin...)
Affinity DataEC50:  140nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014751(3-[1,1-Bis-(4-chloro-phenyl)-ethyl]-pyridine | CHE...)
Affinity DataEC50:  145nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014786(2-[Bis-(4-chloro-phenyl)-methyl]-2H-tetrazole | CH...)
Affinity DataEC50:  150nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014758(Bis-(4-chloro-phenyl)-pyridin-3-yl-methanol | CHEM...)
Affinity DataEC50:  150nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50014801(4-[Bis-(4-chloro-phenyl)-methyl]-pyridine; hydroch...)
Affinity DataEC50:  160nMAssay Description:In vitro Cytochrome P450 19A1 inhibition concentration to decrease aromatization of androstenedione in rat ovarian microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50024522((4-Chloro-phenyl)-(4-fluoro-phenyl)-pyrimidin-5-yl...)
Affinity DataEC50:  180nMAssay Description:In vitro inhibition of cytochrome P450 19A1 by rat ovarian microsomes incubated with [3H]androstenedione and NADPH-generating system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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