Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ec50 data for polymerid = 278
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50: <1nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  5.30nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  30nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  50nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair