Affinity DataEC50: <1nMAssay Description:Dissociation constant for complex with muscarinic acetylcholine receptor M3 of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Dissociation constant for complex with muscarinic acetylcholine receptor M3 of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by Muscarinic M3 receptor)More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at muscarinic M3 receptor in guinea pig trachea assessed as bronchorelaxation activity in presence of propranololMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at muscarinic M3 receptor in guinea pig trachea assessed as bronchorelaxation activity in presence of propranololMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Compound was tested in vitro for the contraction of guinea pig myenteric plexus preparation (mediated by muscarinic acetylcholine receptor M3)More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Compound was tested in vitro for depolarizing response on the rat superior cervical ganglion(mediated by Muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by Muscarinic M3 receptor)More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.11E+3nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.16E+3nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.67E+3nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+3nMAssay Description:In vitro ability of the compound to contract isolated guinea pig ileum was used to estimate M2/M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 6.40E+3nMAssay Description:In vitro ability of the compound to contract isolated guinea pig ileum was used to estimate M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 6.50E+3nMAssay Description:In vitro ability of the compound to contract isolated guinea pig ileum was used to estimate M2/M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 8.60E+3nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 4.49E+4nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 4.64E+4nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+5nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair