Affinity DataEC50: 2.00E+3nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Displacement of [3H]ryanodine from RyR1 calcium channel in sarcoplasmic reticulum assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80E+3nMAssay Description:Displacement of [3H]ryanodine from RyR1 calcium channel in sarcoplasmic reticulum assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.36E+4nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Activation of ryanodine receptor 1 in mouse C2C12 cells assessed as induction of calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.47E+4nMAssay Description:Displacement of [3H]ryanodine from RyR1 calcium channel in sarcoplasmic reticulum assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.06E+4nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]ryanodine from RyR1 calcium channel in sarcoplasmic reticulum assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Displacement of [3H]ryanodine from Ry1R/FKBP12 receptor complex in rabbit sarcoplasmic reticulumMore data for this Ligand-Target Pair