Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ec50 data for polymerid = 50000741,50000742,50002183
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318484(2-((1R,6R)-6-Isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat TRPV2 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50285610(CBV | CHEMBL4170268)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285610(CBV | CHEMBL4170268)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50511105(GWP-42004 | Gwp42004 | O-4394 | THCV | Tetrahydroc...)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463447(CHEMBL4249046)
Affinity DataEC50:  5.80E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463442(CHEMBL4242719)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50532215(CBD-V | CBDV | Cannabidivarin | GWP42006)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50463446(CHEMBL4244422)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol |...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol |...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed