Compile Data Set for Download or QSAR
maximum 50k data
Found 272 of ec50 data for polymerid = 50000827,50007138
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189503(CHEMBL3828298)
Affinity DataEC50:  0.189nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189503(CHEMBL3828298)
Affinity DataEC50:  0.189nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  0.790nMAssay Description:Agonist activity at recombinant human N-terminal epitope tagged/C-terminal eYFP-fused FLAG-tagged GPR84 expressed in Flp-In TREx 293 cell membranes a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human N-terminal epitope tagged/C-terminal eYFP-fused FLAG-tagged GPR84 expressed in Flp-In TREx 293 cell membranes a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189504(CHEMBL3827638)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189505(CHEMBL13302)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50078852(CHEMBL221598)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human GPR84 expressed in HEK293 cells assessed as reduction in forskolin-stimulated cAMP production incubated for 60 mins by HTRF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50511034(CHEMBL4444010)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells co-expressing beta-galactosidase/beta-arrestin2 assessed as inhibition of forskoli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50028344(6-Hexylamino-1H-pyrimidine-2,4-dione | CHEMBL12497...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells assessed as beta-arrestin 2 recruitment measured after 90 mins by beta-galactosida...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50028344(6-Hexylamino-1H-pyrimidine-2,4-dione | CHEMBL12497...)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells co-expressing beta-galactosidase/beta-arrestin2 assessed as inhibition of forskoli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189507(CHEMBL3828303)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189511(CHEMBL3827580)
Affinity DataEC50:  11nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50511013(CHEMBL4538049)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR84 expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP production incubated for 30 mins by lumi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189538(CHEMBL3828708)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GPR84 in mouse bone-marrow-derived neutrophils assessed as stimulation of [35S]GTPgammaS binding incubated for 60 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  16nMAssay Description:Agonist activity at GPR84 in LPS-treated human THP-1 cell membrane assessed as stimulation of [35S]GTPgammaS binding incubated for 60 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189502(CHEMBL3827832)
Affinity DataEC50:  17nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells co-expressing beta-galactosidase/beta-arrestin2 assessed as inhibition of forskoli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189502(CHEMBL3827832)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GPR84 expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP production incubated for 30 mins by lumi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  26nMAssay Description:Agonist activity at GPR84 in LPS-treated mouse RAW 264.7 cell membrane assessed as stimulation of [35S]GTPgammaS binding incubated for 60 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human Galphai2-coupled GPR84 expressed in human Flp-In-T-REx-293 cell membrane assessed as stimulation of [35S]GTPgammaS binding ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse Galphai2-coupled GPR84 expressed in human Flp-In-T-REx-293 cell membrane assessed as stimulation of [35S]GTPgammaS binding ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50556777(CHEMBL4743442)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR84 expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP production incubated for 30 mins by lumi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239172(CHEMBL4088884)
Affinity DataEC50:  41nMAssay Description:Agonist activity at Gi coupled human GPR84 expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 15 mins in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239172(CHEMBL4088884)
Affinity DataEC50:  42nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189510(CHEMBL3827526)
Affinity DataEC50:  49nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239171(CHEMBL4078546)
Affinity DataEC50:  52nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239196(CHEMBL246504)
Affinity DataEC50:  59nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239191(CHEMBL4062512)
Affinity DataEC50:  62nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239194(CHEMBL4101728)
Affinity DataEC50:  80nMAssay Description:Agonist activity at Gi coupled human GPR84 expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 15 mins in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239170(CHEMBL4096571)
Affinity DataEC50:  84nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189508(CHEMBL3828073)
Affinity DataEC50:  88nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50078850(CHEBI:4778 | Embelin)
Affinity DataEC50:  89nMAssay Description:Agonist activity at recombinant human HA-tagged GPR84 stably expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239213(CHEMBL246298)
Affinity DataEC50:  103nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50511034(CHEMBL4444010)
Affinity DataEC50:  104nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells assessed as beta-arrestin 2 recruitment measured after 90 mins by beta-galactosida...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189502(CHEMBL3827832)
Affinity DataEC50:  105nMAssay Description:Agonist activity at recombinant human GPR84 expressed in HEK293 cells co-expressing Gqi5 assessed as increase in myo-[3H]inositol phosphate accumulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239191(CHEMBL4062512)
Affinity DataEC50:  113nMAssay Description:Agonist activity at Gi coupled human GPR84 expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 15 mins in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189502(CHEMBL3827832)
Affinity DataEC50:  114nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells assessed as beta-arrestin 2 recruitment measured after 90 mins by beta-galactosida...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239172(CHEMBL4088884)
Affinity DataEC50:  115nMAssay Description:Agonist activity at GPR84 in LPS-treated human THP-1 cell membrane assessed as stimulation of [35S]GTPgammaS binding incubated for 60 mins by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239218(CHEMBL4104992)
Affinity DataEC50:  129nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  134nMAssay Description:Agonist activity at recombinant human GPR84 stably expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of forskolin-induced cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  139nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  144nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239193(CHEMBL4066454)
Affinity DataEC50:  175nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50239172(CHEMBL4088884)
Affinity DataEC50:  178nMAssay Description:Agonist activity at GPR84 in LPS-treated mouse RAW 264.7 cell membrane assessed as stimulation of [35S]GTPgammaS binding incubated for 60 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239171(CHEMBL4078546)
Affinity DataEC50:  187nMAssay Description:Agonist activity at Gi coupled human GPR84 expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 15 mins in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239194(CHEMBL4101728)
Affinity DataEC50:  199nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50078850(CHEBI:4778 | Embelin)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant human N-terminal epitope tagged/C-terminal eYFP-fused FLAG-tagged GPR84 expressed in Flp-In TREx 293 cell membranes a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189549(CHEMBL3827756)
Affinity DataEC50:  213nMAssay Description:Agonist activity at recombinant human GPR84 stably expressed in HEK293 cells co-expressing Galpha16 assessed as increase in intracellular calcium mob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50189553(CHEMBL3827763)
Affinity DataEC50:  231nMAssay Description:Agonist activity at GPR84 (unknown origin) expressed in HEK293 cells coexpressing Galpha16 protein by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239195(CHEMBL4096406)
Affinity DataEC50:  250nMAssay Description:Positive allosteric modulation of recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 assessed as increase in [3H]PS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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