Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ec50 data for polymerid = 50005943
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301356(CHEMBL585927 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in osteocalcin levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301356(CHEMBL585927 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in alkaline phosphatase levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301364(CHEMBL570380 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in alkaline phosphatase levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301364(CHEMBL570380 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301364(CHEMBL570380 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in osteocalcin levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 2-beta(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50301356(CHEMBL585927 | N-(5-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataEC50:  10nMAssay Description:Inhibition of mouse Pyk2 in MC3TC3 cells assessed as increase in calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed