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Found 5 of ec50 data for polymerid = 50006059,50006915
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526580(CHEMBL4549036)
Affinity DataEC50:  300nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  780nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526578(CHEMBL4468490)
Affinity DataEC50:  2.06E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526579(CHEMBL4442766)
Affinity DataEC50:  2.36E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM81289(Adenosine 3',5'-cyclic monophosphate sodiu...)
Affinity DataEC50:  3.87E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed