Compile Data Set for Download or QSAR
maximum 50k data
Found 118 of ec50 data for polymerid = 5550,49000265,49000266,50002396,50004273,50004685
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159153(CHEMBL3787243)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159153(CHEMBL3787243)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159151(CHEMBL3786145)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159151(CHEMBL3786145)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159152(CHEMBL3786986)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159152(CHEMBL3786986)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159154(CHEMBL3787379)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50159154(CHEMBL3787379)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ assessed as induction of intracellular Ca2+ mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50518037(CHEMBL4542269)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human AT1 receptor assessed as increase in beta-arrestin recruitment by chemiluminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50518053(CHEMBL4438122)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human AT1 receptor assessed as increase in beta-arrestin recruitment by chemiluminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282221(2-Ethyl-4-hydroxy-5-phenyl-7-[2'-(1H-tetrazol-5-yl...)
Affinity DataEC50:  90nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataEC50:  350nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282222(7-Ethoxy-4-hydroxy-3-phenyl-1-[2'-(1H-tetrazol-5-y...)
Affinity DataEC50:  500nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282218(4-Hydroxy-7-methylsulfanyl-3-phenyl-1-[2'-(1H-tetr...)
Affinity DataEC50:  600nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282219(4-Hydroxy-7-methyl-3-phenyl-1-[2'-(1H-tetrazol-5-y...)
Affinity DataEC50:  1.25E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282215(4-Hydroxy-3-phenyl-1-[2'-(1H-tetrazol-5-yl)-biphen...)
Affinity DataEC50:  1.25E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282217(4-Hydroxy-3-phenyl-1-[2'-(1H-tetrazol-5-yl)-biphen...)
Affinity DataEC50:  1.70E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282216(4'-(7-Ethoxy-4-hydroxy-2-oxo-3-phenyl-2H-quinolin-...)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282223(4-Hydroxy-7-methoxy-3-phenyl-1-[2'-(1H-tetrazol-5-...)
Affinity DataEC50:  2.20E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type AGTR1 receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50499311(CHEMBL3736156)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type AGTR1 receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50499310(CHEMBL3736433)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type AGTR1 receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50028423(CHEMBL3355127)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50028420(CHEMBL3355137)
Affinity DataEC50:  5.50E+3nMAssay Description:Agonist activity at AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282214(7-Hydroxy-6-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphen...)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM51796((5Z)-5-[(2Z)-2-(3-ethyl-4,5-diphenyl-1,3-thiazol-2...)
Affinity DataEC50:  7.44E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282220(4'-(4-Hydroxy-7-methoxy-2-oxo-3-phenyl-2H-quinolin...)
Affinity DataEC50:  9.50E+3nMAssay Description:Inhibition of [125I]-AII binding to angiotensin II receptor of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50183341(CHEMBL3817879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544720(CHEMBL4632564)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544728(CHEMBL4641474)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544736(CHEMBL4647853)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544735(CHEMBL4640815)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544729(CHEMBL4647391)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544744(CHEMBL4647996)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544742(CHEMBL4647910)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544721(CHEMBL4644803)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544749(CHEMBL4640653)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50544733(CHEMBL4640390)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human AGTR1 stably expressed in CHO cells assessed as increase in intracellular calcium mobilization measured at 1 sec intervals ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50571385(CHEMBL4875417)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Galphaq16-fused human AGTR1 expressed in CHO cells assessed as stimulation of Ca2+ mobilization incubated for 1 hr by Calcium 5-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM66953(4-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-N-[3-(...)
Affinity DataEC50:  5.78E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76097(2-(3-Cyclohexyl-3H-imidazo[4,5-b]pyridin-2-ylsulfa...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76098(3-({[1-(1-Benzyl-1H-tetrazol-5-yl)-propyl]-furan-2...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76099(3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-oxolanylm...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76100(3-[[[1-(1-cyclohexyl-1,2,3,4-tetrazol-5-yl)-2-meth...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76101(3-[[1-(1-benzyltetrazol-5-yl)propyl-(oxolan-2-ylme...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM76102(6-Methoxy-3-{[{1-[1-(2-methoxy-ethyl)-1H-tetrazol-...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM38416(4-(2-furyl)-6,8-dimethyl-2-piperidin-1-ylpyrimido[...)
Affinity DataEC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego) Ne...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
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