Compile Data Set for Download or QSAR
maximum 50k data
Found 438 of ec50 data for polymerid = 5923,8490
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50526270(CHEMBL4554474)
Affinity DataEC50:  143nMAssay Description:Activation of dephosphorylated IRE1alpha (G547 to L977 residues) (unknown origin)-dependent cleavage of FAM-labeled stem-loop RNA containing the XBP1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111358(US8614253, 29-18 | US9241942, 29-18)
Affinity DataEC50:  1.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111346(US8614253, 29-6 | US8614253, 42-4 | US9241942, 42-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111346(US8614253, 29-6 | US8614253, 42-4 | US9241942, 42-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111359(US8614253, 29-19 | US9241942, 29-19 | US9493435, 1...)
Affinity DataEC50:  3.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111316(US8614253, 43-76 | US9241942, 27-76)
Affinity DataEC50:  3.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111343(US8614253, 29-3 | US9241942, 29-3)
Affinity DataEC50:  4.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111342(US8614253, 29-2 | US9241942, 29-2)
Affinity DataEC50:  5.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111368(US8614253, 32-4 | US9241942, 32-4 | US9493435, 168)
Affinity DataEC50:  5.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111344(US8614253, 29-4 | US9241942, 29-4)
Affinity DataEC50:  5.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111382(US8614253, 34-1 | US9241942, 34-1)
Affinity DataEC50:  7.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111347(US8614253, 29-7 | US9241942, 29-7)
Affinity DataEC50:  7.00E+3nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111341(US8614253, 29-1 | US9241942, 29-1)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111345(US8614253, 29-5 | US9241942, 29-5)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111348(US8614253, 29-8 | US9241942, 29-8)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111357(US8614253, 29-17 | US9241942, 29-17)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111364(US8614253, 31-2 | US8614253, 32-14 | US8614253, 42...)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111384(US8614253, 34-3 | US9241942, 34-3)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM111428(US8614253, 42-3 | US9241942, 42-3)
Affinity DataEC50:  1.00E+4nMAssay Description:Initial cell-based XBP-1 mRNA splicing assays confirmed IRE-1α inhibition with several potent 5-bromo and 6 bromo o-vanillins. HEK293 cells were...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160334(US9040714, 1 | US9693992, 1)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160335(US9040714, 2 | US9693992, 2)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM51439(BDBM160336 | US9040714, 116 | US9693992, 116)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160337(US9040714, 4 | US9693992, 4)
Affinity DataIC50: <100nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160338(US9040714, 5 | US9693992, 5)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160339(US9040714, 6 | US9693992, 6)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160340(US9040714, 7 | US9693992, 7)
Affinity DataIC50: <100nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160341(US9040714, 8 | US9693992, 8)
Affinity DataIC50: >1.00E+4nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160342(US9040714, 9 | US9693992, 9)
Affinity DataIC50: <1.00E+3nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160343(US9040714, 10 | US9693992, 10)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160344(US9040714, 11 | US9693992, 11)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160345(US9040714, 12 | US9693992, 12)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160346(US9040714, 13 | US9693992, 13)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160347(US9040714, 14 | US9693992, 14)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM65602(US9693992, 15)
Affinity DataEC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160348(US9040714, 16 | US9693992, 16)
Affinity DataIC50: <100nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160349(US9040714, 17 | US9693992, 17)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160350(US9040714, 18 | US9693992, 18)
Affinity DataIC50: <1.00E+3nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160351(US9040714, 19 | US9693992, 19)
Affinity DataIC50: >1.00E+3nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160352(US9040714, 20 | US9693992, 20)
Affinity DataIC50: <1.00E+3nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160353(US9040714, 21 | US9693992, 21)
Affinity DataIC50: <100nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160354(US9040714, 22 | US9693992, 22)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160355(US9040714, 23 | US9693992, 23)
Affinity DataIC50: <1.00E+3nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160356(US9040714, 24 | US9693992, 24)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160357(US9040714, 25 | US9693992, 25)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160358(US9040714, 26 | US9693992, 26)
Affinity DataIC50: <1.00E+3nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160359(US9040714, 27 | US9693992, 27)
Affinity DataIC50: <100nM EC50: <1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160360(US9040714, 28 | US9693992, 28)
Affinity DataIC50: <1.00E+4nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160365(US9040714, 33 | US9693992, 33)
Affinity DataIC50: <1.00E+4nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160366(US9040714, 34 | US9693992, 34)
Affinity DataIC50: <1.00E+4nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM160367(US9040714, 35 | US9693992, 35)
Affinity DataIC50: <100nM EC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) obtained from a 500 ml baculovirus-infected ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
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