TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 4.5nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg
Curated by ChEMBL
University Of Halle-Wittenberg
Curated by ChEMBL
Affinity DataEC50: >2.20E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair