Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ec50 data for polymerid = 7527
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542677(CHEMBL4637446)
Affinity DataEC50:  1.10nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542678(CHEMBL4636474)
Affinity DataEC50:  1.70nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542676(CHEMBL4633668)
Affinity DataEC50:  4.5nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50581535(CHEMBL5091040)
Affinity DataEC50:  130nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50581544(CHEMBL5086475)
Affinity DataEC50:  600nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50581547(CHEMBL5081349)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50581545(CHEMBL5084902)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50581546(CHEMBL5084416)
Affinity DataEC50: >2.20E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed