Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ec50 data for polymerid = 9635
TargetN-lysine methyltransferase KMT5A(Homo sapiens (Human))
The Center For Combinatorial Chemistry And Drug Discovery Of Jilin University

Curated by ChEMBL
LigandPNGBDBM50075100(CHEMBL3414625)
Affinity DataEC50: <1.00E+3nMAssay Description:Inhibition of SETD8 in HEK293T cells assessed as reduction in H4K20me level after 2 to 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-lysine methyltransferase KMT5A(Homo sapiens (Human))
The Center For Combinatorial Chemistry And Drug Discovery Of Jilin University

Curated by ChEMBL
LigandPNGBDBM50106497(6-Chloro-7-(2-morpholin-4-yl-ethylamino)-quinoline...)
Affinity DataEC50: <5.00E+3nMAssay Description:Inhibition of SETD8 in HEK293T cells assessed as reduction in H4K20me level after 2 to 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-lysine methyltransferase KMT5A(Homo sapiens (Human))
The Center For Combinatorial Chemistry And Drug Discovery Of Jilin University

Curated by ChEMBL
LigandPNGBDBM50075099(CHEMBL580421 | TCMDC-124224)
Affinity DataEC50: <5.00E+3nMAssay Description:Inhibition of SETD8 in HEK293T cells assessed as reduction in H4K20me level after 2 to 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed