Compile Data Set for Download or QSAR
maximum 50k data
Found 63 of ic50 data for polymerid = 2445,50000355,50002089
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  0.5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  180nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  290nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  300nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibitory concentration against adipocyte-derived leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50:  3.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50046329(3-Amino-4-(4-benzyloxy-phenyl)-2-oxo-butyric acid ...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50046316(2-Amino-3-(4-benzyloxy-phenyl)-propane-1-thiol | C...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534077(CHEMBL4464704)
Affinity DataIC50:  6.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534070(CHEMBL4454667)
Affinity DataIC50:  6.83E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534074(CHEMBL4468968)
Affinity DataIC50:  6.93E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534069(CHEMBL4473220)
Affinity DataIC50:  7.68E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50046321(3-Amino-4-(4-benzyloxy-phenyl)-2-hydroxy-butyric a...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23977((3Z)-3-[(2-phenylethoxy)imino]-1,2,3,4-tetrahydron...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23980((3Z)-3-{[(5-phenylpentyl)oxy]imino}-1,2,3,4-tetrah...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336496(2-aminocycloheptanone hydrochloride | CHEMBL166862...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50046314(3-Amino-4-(4-benzyloxy-phenyl)-2-oxo-butyric acid ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23979((3Z)-3-[(4-phenylbutoxy)imino]-1,2,3,4-tetrahydron...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50051495((S)-2-[(S)-2-(2-Hydroxy-acetyl)-pyrrolidine-1-carb...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of proline iminopeptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534072(CHEMBL4455383)
Affinity DataIC50:  1.11E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50:  1.20E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534078(CHEMBL4557950)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534081(CHEMBL4460083)
Affinity DataIC50:  1.63E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534071(CHEMBL4563759)
Affinity DataIC50:  3.79E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534080(CHEMBL4576374)
Affinity DataIC50:  4.09E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  4.50E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
National Institute Of Public Health-National Institute Of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534073(CHEMBL4537106)
Affinity DataIC50:  7.81E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336493(1-Aminoindan-2-one, hydrochloride | CHEMBL1668624)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336494(6-amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one,...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336495(7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one,...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23988(2-amino-1,2,3,4-tetrahydroisoquinolin-3-one | N-Su...)
Affinity DataIC50:  1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336497(7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM50336499(CHEMBL1668630 | cis-7-amino-6,7,8,9-tetrahydro-5H-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23987(2-hydroxy-1,2,3,4-tetrahydroisoquinolin-3-one | CH...)
Affinity DataIC50: >1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23986(3,4-dihydro-1H-2-benzothiopyran-3-one | isothiochr...)
Affinity DataIC50: >1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23985(3,4-dihydro-1H-2-benzopyran-3-one | isochromanone,...)
Affinity DataIC50: >1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23984(3-amino-1,2,3,4-tetrahydronaphthalene-2-phosphonic...)
Affinity DataIC50: >1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Bos taurus (bovine))
Enscmu

LigandPNGBDBM23982(1-(3-amino-1,2,3,4-tetrahydronaphthalen-2-yl)ethan...)
Affinity DataIC50: >1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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