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Found 37 of ic50 data for polymerid = 49000244
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against beta-1 adrenergic receptor in guinea pig atria is determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036835(1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol |...)
Affinity DataIC50:  115nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017383(9a-Methoxy-5,6,7,8,9,9a-hexahydro-4bH-benzo[a]azul...)
Affinity DataIC50:  160nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataIC50:  190nMAssay Description:Tested for beta1-adrenergic blocking effect by measuring the ability to inhibit the positive inotropic effect of isoproterenol on the isolated right ...More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataIC50:  320nMAssay Description:Tested for beta-2-adrenergic blocking effect by measuring the ability to inhibit the relaxing effect of epinephrine on the isolated tracheal muscle o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017385(9a-Hydroxy-5,6,7,8,9,9a-hexahydro-4bH-benzo[a]azul...)
Affinity DataIC50:  340nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017396(7-Fluoro-9a-methoxy-1,2,3,4,4a,9a-hexahydro-fluore...)
Affinity DataIC50:  830nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017390(9a-(2-Hydroxy-ethoxy)-1,2,3,4,4a,9a-hexahydro-fluo...)
Affinity DataIC50:  850nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017395(9a-Hydroxy-5,6,7,8,9,9a-hexahydro-4bH-benzo[a]azul...)
Affinity DataIC50:  890nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017388(9a-Methoxy-1,2,3,4,4a,9a-hexahydro-fluoren-9-one O...)
Affinity DataIC50:  1.20E+3nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50289372((S)-1,1-Difluoro-3-isopropylamino-1-[4-(2-methoxy-...)
Affinity DataIC50:  1.35E+3nMAssay Description:Tested for beta-1-adrenergic blocking effect by measuring the ability to inhibit the positive inotropic effect of isoproterenol on the isolated right...More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50289372((S)-1,1-Difluoro-3-isopropylamino-1-[4-(2-methoxy-...)
Affinity DataIC50:  2.15E+3nMAssay Description:Tested for beta-2-adrenergic blocking effect by measuring the ability to inhibit the relaxing effect of epinephrine on the isolated tracheal muscle o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017387(9a-Hydroxy-1,2,3,4,4a,9a-hexahydro-fluoren-9-one O...)
Affinity DataIC50:  2.80E+3nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017392(9a-Methoxy-5,6,7,8,9,9a-hexahydro-4bH-benzo[a]azul...)
Affinity DataIC50:  3.00E+3nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50041914(1-Aminomethyl-isochroman-6,7-diol | CHEMBL105383)
Affinity DataIC50:  6.76E+3nMAssay Description:Inhibitory activity against beta-1 adrenergic receptor in guinea pig atria is determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036842(3-tert-Butylamino-2-hydroxy-propionaldehyde O-prop...)
Affinity DataIC50:  8.32E+3nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017391(9a-(2-Hydroxy-ethoxy)-5,6,7,8,9,9a-hexahydro-4bH-b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017381(7-Fluoro-9a-methoxy-1,2,3,4,4a,9a-hexahydro-fluore...)
Affinity DataIC50: >1.00E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017389(13a-Methoxy-5,6,7,8,9,10,11,12,13,13a-decahydro-4b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017380(9a-(2-Hydroxy-ethoxy)-5,6,7,8,9,9a-hexahydro-4bH-b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017394(9a-Methoxy-1,2,3,4,4a,9a-hexahydro-fluoren-9-one O...)
Affinity DataIC50: >1.00E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017384(9a-Methoxy-1,2,3,4,4a,9a-hexahydro-fluoren-9-one O...)
Affinity DataIC50:  1.20E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036839(2-Hydroxy-3-isopropylamino-propionaldehyde O-ethyl...)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017379(9a-Methoxy-5,6,7,8,9,9a-hexahydro-4bH-benzo[a]azul...)
Affinity DataIC50:  1.30E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036838(Acetaldehyde O-(3-tert-butylamino-2-hydroxy-propyl...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036841(3-tert-Butylamino-2-hydroxy-propionaldehyde O-ethy...)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036836(CHEMBL38114 | Propionaldehyde O-(2-hydroxy-3-isopr...)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036837(2-Hydroxy-3-isopropylamino-propionaldehyde O-propy...)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017386(7-Fluoro-9a-methoxy-1,2,3,4,4a,9a-hexahydro-fluore...)
Affinity DataIC50:  1.90E+4nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036840(CHEMBL38033 | Propionaldehyde O-(3-tert-butylamino...)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036843(Acetaldehyde O-(2-hydroxy-3-isopropylamino-propyl)...)
Affinity DataIC50:  3.02E+4nMAssay Description:Inhibitory concentration against beta-1-adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50041915(1-(Isopropylamino-methyl)-isochroman-6,7-diol | CH...)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibitory activity against beta-1 adrenergic receptor in guinea pig atria is determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50010891(1-Aminomethyl-isochroman-5,6-diol | 1-Aminomethyl-...)
Affinity DataIC50:  6.61E+4nMAssay Description:Inhibitory activity against beta-1 adrenergic receptor in guinea pig atria is determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017393(9a-Hydroxy-1,2,3,4,4a,9a-hexahydro-fluoren-9-one O...)
Affinity DataIC50: >1.00E+5nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017378(9a-(2-Hydroxy-ethoxy)-1,2,3,4,4a,9a-hexahydro-fluo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017382(13a-Methoxy-5,6,7,8,9,10,11,12,13,13a-decahydro-4b...)
Affinity DataIC50: >1.00E+5nMAssay Description:Beta-1 adrenergic receptor blocking was assessed from 50% inhibition of the isoproterenol submaximal response on isolated Guinea pig atria(IA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50041913(1-(Isopropylamino-methyl)-isochroman-5,6-diol | CH...)
Affinity DataIC50: <3.16E+5nMAssay Description:Inhibitory activity against beta-1 adrenergic receptor in guinea pig atria is determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed