Compile Data Set for Download or QSAR
maximum 50k data
Found 23 of ic50 data for polymerid = 49000285
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264141(1-Benzyl-1H-benzoimidazole-2-carboxylic acid {2-[6...)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  2.80nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50203200((R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((R)-...)
Affinity DataIC50:  4nMAssay Description:Antagonistic activity at rat bradykinin B1 receptor assessed as effect on DAK-mediated calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50370213(CHEMBL1744083)
Affinity DataIC50:  7.25nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264368(1-benzyl-N-ethyl-N-(2-(4-(1-methylpiperidin-4-yl)p...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381270(CHEMBL2018868)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381265(CHEMBL2018873)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264370(1-benzyl-N-(2-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50370216(CHEMBL1744084)
Affinity DataIC50:  24.2nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50370217(CHEMBL1744085)
Affinity DataIC50:  27nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381271(CHEMBL2018867)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381266(CHEMBL2018872)
Affinity DataIC50:  42nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381273(CHEMBL2018874)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381267(CHEMBL2018871)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381269(CHEMBL2018869)
Affinity DataIC50:  52nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50370215(CHEMBL1744082)
Affinity DataIC50:  59nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50381268(CHEMBL2018870)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264298(CHEMBL490201 | N-(2-((4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataIC50:  155nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50156455((R)-N-(4-(4,5-dihydro-1H-imidazol-2-yl)phenethyl)-...)
Affinity DataIC50:  164nMAssay Description:Inhibition of rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264140(CHEMBL492211 | N-(2-((4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataIC50:  345nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264369(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50:  396nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264296(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50:  417nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed