Compile Data Set for Download or QSAR
maximum 50k data
Found 52 of ic50 data for polymerid = 50000654,50000655,50004578,50006269
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  1.29nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  45.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414658(CHEMBL559048)
Affinity DataIC50:  58.9nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414645(CYASTERONE)
Affinity DataIC50:  61.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414646(INOKOSTERONE)
Affinity DataIC50:  91.2nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50226672(CHEMBL255034 | makisterone A)
Affinity DataIC50:  112nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414659(CHEMBL564892)
Affinity DataIC50:  324nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414652(CHEMBL559941)
Affinity DataIC50:  794nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  900nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488465(CHEMBL2286413)
Affinity DataIC50:  2.24E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414651(ECDYSONE)
Affinity DataIC50:  2.57E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326770(4-isobutyl-5-methylene-2-oxo-1-(2,4,5-trichlorophe...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326767(4-butyl-1-(2-tert-butyl-5-chlorophenyl)-5-methylen...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326755(1-(2,5-di-tert-butylphenyl)-4-methyl-5-methylene-2...)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326760(4-ethyl-5-methylene-2-oxo-1-(2,4,5-trichlorophenyl...)
Affinity DataIC50:  7.25E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326765(4-butyl-1-(3-chloro-2-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  8.30E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326758(1-(4-tert-butyl-2,5-dichlorophenyl)-4-methyl-5-met...)
Affinity DataIC50:  8.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488464(CHEMBL2286419)
Affinity DataIC50:  8.91E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414655(CHEMBL560796)
Affinity DataIC50:  9.55E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326759(1-(2-tert-butyl-5-chlorophenyl)-4-ethyl-5-methylen...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326773(1-cyclohexyl-5-methylene-2-oxo-4-phenyl-2,5-dihydr...)
Affinity DataIC50:  1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326766(4-butyl-1-(5-chloro-2-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488463(CHEMBL2285681)
Affinity DataIC50:  1.35E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414657(CHEMBL562711)
Affinity DataIC50:  1.45E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488437(CHEMBL2286416)
Affinity DataIC50:  1.48E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326761(1-(2-tert-butylphenyl)-4-isopropyl-5-methylene-2-o...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326774(3-benzoyl-4-methyl-5-methylene-1-(3-(trifluorometh...)
Affinity DataIC50:  1.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326756(1-(2,6-diisopropylphenyl)-4-methyl-5-methylene-2-o...)
Affinity DataIC50:  2.35E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488438(CHEMBL2286414)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488477(CHEMBL2286417)
Affinity DataIC50:  2.69E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326757(1-(3,5-dichlorophenyl)-4-methyl-5-methylene-2-oxo-...)
Affinity DataIC50:  2.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488448(CHEMBL2286411)
Affinity DataIC50:  2.82E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326769(4-butyl-1-(2-ethyl-6-methylphenyl)-5-methylene-2-o...)
Affinity DataIC50:  3.30E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414660(CHEMBL564474)
Affinity DataIC50:  3.89E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414649(CHEMBL561275)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414647(CHEMBL560194)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326762(1-(2-tert-butyl-4-chlorophenyl)-4-isopropyl-5-meth...)
Affinity DataIC50:  4.20E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326763(4-isopropyl-1-(2-isopropyl-6-methylphenyl)-5-methy...)
Affinity DataIC50:  4.70E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488462(CHEMBL2286415)
Affinity DataIC50:  4.79E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326754(4-methyl-5-methylene-2-oxo-1-(2-(trifluoromethyl)p...)
Affinity DataIC50:  4.80E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326772(1-(2-isopropyl-6-methylphenyl)-5-methylene-2-oxo-4...)
Affinity DataIC50:  5.50E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326768(4-butyl-1-(2-chloro-6-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  5.60E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488447(CHEMBL2286412)
Affinity DataIC50:  6.76E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414653(CHEMBL558256)
Affinity DataIC50:  8.91E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326771(4-isobutyl-1-mesityl-5-methylene-2-oxo-2,5-dihydro...)
Affinity DataIC50:  1.75E+5nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414648(CHEMBL559545)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414650(CHEMBL550600)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414654(CHEMBL560139)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414656(CHEMBL558652)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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