Compile Data Set for Download or QSAR
maximum 50k data
Found 54 of ic50 data for polymerid = 50001894
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50449890(CHEMBL4161876)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50449891(CHEMBL4174756)
Affinity DataIC50:  13nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50520631(Ametantrone)
Affinity DataIC50:  30nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50449889(CHEMBL4160802)
Affinity DataIC50:  32nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50449888(CHEMBL4172196)
Affinity DataIC50:  81nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50449887(CHEMBL4169404)
Affinity DataIC50:  110nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50547613(CHEMBL4751362)
Affinity DataIC50:  130nMAssay Description:Inhibition of Topoisomerase II beta (unknown origin) relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473498(CHEMBL157831 | Ro-616653)
Affinity DataIC50:  157nMAssay Description:Antibacterial activity against Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473498(CHEMBL157831 | Ro-616653)
Affinity DataIC50:  157nMAssay Description:Antibacterial activity against Micrococcus luteus DNA gyrase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473499(BAY-507950 | CHEMBL156813)
Affinity DataIC50:  326nMAssay Description:Antibacterial activity against Micrococcus luteus DNA gyrase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229974(CHEMBL178077)
Affinity DataIC50:  452nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473499(BAY-507950 | CHEMBL156813)
Affinity DataIC50:  489nMAssay Description:Antibacterial activity against Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50458474(CHEMBL4213218)
Affinity DataIC50:  580nMAssay Description:Inhibition of human topoisomerase-2B after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  603nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473497(BAY-507952 | CHEMBL157769)
Affinity DataIC50:  625nMAssay Description:Antibacterial activity against Micrococcus luteus DNA gyrase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229967(CHEMBL263944)
Affinity DataIC50:  666nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229969(CHEMBL554645)
Affinity DataIC50:  727nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  727nMAssay Description:Inhibition of Topoisomerase II beta (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473497(BAY-507952 | CHEMBL157769)
Affinity DataIC50:  781nMAssay Description:Antibacterial activity against Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  790nMAssay Description:Inhibition of human topoisomerase-2B after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229970(CHEMBL367876)
Affinity DataIC50:  796nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50458475(CHEMBL4205327)
Affinity DataIC50:  860nMAssay Description:Inhibition of human topoisomerase-2B after 2 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  905nMAssay Description:Gyrase inhibitory activity against Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229972(CHEMBL174721)
Affinity DataIC50:  929nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50520632(CHEMBL4553471)
Affinity DataIC50:  1.06E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50520634(CHEMBL4575796)
Affinity DataIC50:  1.15E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229966(DESMETHYL-OFLOXACIN | Desmethyl-Ofloxacin (5%))
Affinity DataIC50:  1.69E+3nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50229965(CHEMBL174892)
Affinity DataIC50:  2.58E+3nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50227628(CHEMBL47311)
Affinity DataIC50:  2.67E+3nMAssay Description:Gyrase inhibitory activity against Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM87351(Amsacrine hydrochloride | CHEMBL43 | MLS002153376 ...)
Affinity DataIC50:  2.76E+3nMAssay Description:Inhibition of human topoisomerase-2B after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataIC50:  2.76E+3nMAssay Description:Gyrase inhibitory activity against Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50045004(9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-ox...)
Affinity DataIC50:  2.76E+3nMAssay Description:Gyrase inhibitory activity against Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50586362(CHEMBL5083245)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human TOP2B assessed as reduction in relaxation of supercoiled DNA using kDNA as substrate incubated for 30 minMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human topoisomerase-2B after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human topoisomerase 2beta after 2 hrs at 37 degC by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50520633(CHEMBL4448353)
Affinity DataIC50:  4.34E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50520636(CHEMBL4467805)
Affinity DataIC50:  5.25E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition effect on Escherichia coli Wild Type DNA gyrase Supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50464488(CHEMBL4278922)
Affinity DataIC50:  9.29E+3nMAssay Description:Inhibition of human topoisomerase 2beta after 2 hrs at 37 degC by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50135927(7-(4-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxazolid...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibitory concentration against Escherichia coli by Escherichia coli DNA gyrase gel-based supercoil assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50586360(ADR-529 | CHEBI:50223 | Cardioxane | DEXRAZOXANE |...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human TOP2B assessed as reduction in relaxation of supercoiled DNA using kDNA as substrate incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50473500(CHEMBL158264)
Affinity DataIC50:  6.25E+4nMAssay Description:Antibacterial activity against Micrococcus luteus DNA gyrase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50:  7.15E+4nMAssay Description:Inhibition of Escherichia coli Quinolone resistant gyrase Supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50366305(CHEBI:70328 | CHEMBL445599)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human topoisomerase 2beta-mediated relaxation of supercoiled pSG483 DNA after 30 mins by ethidium bromide staining based agarose gel el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50471425(CHEMBL110041)
Affinity DataIC50:  1.21E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50554356(CHEMBL4758733)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of recombinant wild-type human topoisomerase 2beta expressed in Saccharomyces cerevisiae using supercoiled pBR322 DNA as substrate measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50471426(CHEMBL110367)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM21691(1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridi...)
Affinity DataIC50:  2.23E+5nMAssay Description:Inhibition of supercoiling activity of DNA gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Port Said University

Curated by ChEMBL
LigandPNGBDBM50586361(CHEMBL5076925)
Affinity DataIC50:  5.05E+5nMAssay Description:Inhibition of human TOP2B assessed as reduction in relaxation of supercoiled DNA using kDNA as substrate incubated for 30 minMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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