Compile Data Set for Download or QSAR
maximum 50k data
Found 37 of ic50 data for polymerid = 843,50007353
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)
Affinity DataIC50:  1nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)
Affinity DataIC50:  2nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235348(CHEMBL4078988)
Affinity DataIC50:  3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235346(CHEMBL4102518)
Affinity DataIC50:  8nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235347(CHEMBL4078246)
Affinity DataIC50:  10nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235349(CHEMBL4065402)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235336(CHEMBL4085238)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235354(CHEMBL4069161)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235344(CHEMBL4086832)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235345(CHEMBL4105278)
Affinity DataIC50:  24nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235340(CHEMBL4101626)
Affinity DataIC50:  26nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235355(CHEMBL4081027)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50246253(4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-(me...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Cyclin A/CDK2More data for this Ligand-Target Pair
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50117488(CHEMBL217362 | H-His-Ala-Lys-Arg-Arg-Leu-Ile-Phe-N...)
Affinity DataIC50:  50nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235356(CHEMBL4097571)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235353(CHEMBL4090226)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235332(CHEMBL4094205)
Affinity DataIC50:  290nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378828(CHEMBL1241134)
Affinity DataIC50:  530nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235357(CHEMBL4089837)
Affinity DataIC50:  580nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378830(CHEMBL1241136)
Affinity DataIC50:  590nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378815(CHEMBL1241137)
Affinity DataIC50:  680nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50:  830nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM5530(2-Anilino-6-cyclohexylmethoxypurine | 6-(cyclohexy...)
Affinity DataIC50:  970nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235339(CHEMBL4073211)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378817(CHEMBL1241139)
Affinity DataIC50:  5.60E+3nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235351(CHEMBL4102300)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235330(CHEMBL4081980)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235352(CHEMBL4084337)
Affinity DataIC50:  8.90E+3nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378816(CHEMBL1241138)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235358(CHEMBL4072216)
Affinity DataIC50:  1.60E+4nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235333(CHEMBL4066675)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50378829(CHEMBL1241135)
Affinity DataIC50:  2.10E+4nMAssay Description:Binding affinity to Cyclin A by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235331(CHEMBL4099986)
Affinity DataIC50:  2.84E+4nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235338(CHEMBL4072170)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed