Affinity DataKd: 3nMpH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.710nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.30nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.730nMAssay Description:Binding of [3H]-CPX to A1 adenosine receptor of DDT1 MF-2 (DDT) cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.30nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.790nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.740nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.280nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.05 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.810nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.310nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.340nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.710nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.270nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.1 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.320nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.260nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.05 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.1 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.460nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
Affinity DataKd: 0.75nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
Affinity DataKd: 4.60E+3nMAssay Description:Affinity for adenosine A1 receptor in CHO membranesMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair