Compile Data Set for Download or QSAR
maximum 50k data
Found 181 of kd data for polymerid = 2129
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKd:  3nMpH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120221(4-[5-(8-Bicyclo[2.2.1]hept-2-yl-2,6-dioxo-1-propyl...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120223(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.400nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039674(Bromo-acetic acid 3-(2,6-dioxo-1,3-dipropyl-2,3,6,...)
Affinity DataKd:  0.710nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039678(8-cyclopentyl-1,3-di[3-(4-fluorosulfonylphenylcarb...)
Affinity DataKd:  0.820nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039696(3-Fluorosulfonyl-benzoic acid 3-(2,6-dioxo-1,3-dip...)
Affinity DataKd:  1.30nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039677(4-[3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  1.80nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039697(Bromo-acetic acid 2-(8-cyclopentyl-2,6-dioxo-1-pro...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039680(8-(2,5-Dioxo-2,5-dihydro-pyrrol-1-ylmethyl)-1,3-di...)
Affinity DataKd:  0.730nMAssay Description:Binding of [3H]-CPX to A1 adenosine receptor of DDT1 MF-2 (DDT) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039684(2-Bromo-N-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahyd...)
Affinity DataKd:  1.30nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039689(3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  0.790nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039685(3-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039691(3-[3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.860nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039695(Bromo-acetic acid 3-(8-cyclopentyl-2,6-dioxo-1-pro...)
Affinity DataKd:  1.5nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039688(4-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.740nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039682(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.280nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.05 nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 5 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095603(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.810nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.310nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.340nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.710nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.270nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.1 nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095606(4-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahy...)
Affinity DataKd:  0.320nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.260nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.05 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095605(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.240nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.1 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50024563(CHEMBL3330574)
Affinity DataKd:  0.460nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50080550((2-Amino-4,5-dimethyl-thiophen-3-yl)-(3-trifluorom...)
Affinity DataKd:  0.75nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50080540((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataKd:  4.60E+3nMAssay Description:Affinity for adenosine A1 receptor in CHO membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083560(CHEMBL3423400)
Affinity DataKd:  1.20E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083559(CHEMBL3423401)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083509(CHEMBL3423402)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083558(CHEMBL3423403)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083555(CHEMBL3423404)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083554(CHEMBL3423405)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083551(CHEMBL3423406)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083550(CHEMBL3423407)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083546(CHEMBL3423408)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50083544(CHEMBL3423409)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor (unknown origin) expressed in sheep striatum membranes after 2 hrs by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50214409((6aR,9R)-N-((S)-1-((S)-1-((S)-2-carbamoylindolin-1...)
Affinity DataKd:  100nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50253852((2-amino-4-((4-methylpiperazin-1-yl)methyl)thiophe...)
Affinity DataKd:  1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50253308((2-amino-4-((4-(pyrimidin-2-yl)piperazin-1-yl)meth...)
Affinity DataKd:  1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50253307((2-amino-4-((4-(pyridin-2-yl)piperazin-1-yl)methyl...)
Affinity DataKd:  1.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50253928((2-amino-4-((4-(4-(trifluoromethyl)phenyl)piperazi...)
Affinity DataKd:  1.90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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