Compile Data Set for Download or QSAR
maximum 50k data
Found 32 of kd data for polymerid = 326,4332
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKd:  1.5nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407340(CHEMBL1790310)
Affinity DataKd:  3.16E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50403724(CHEMBL2110297)
Affinity DataKd:  5.34E+3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407343(CHEMBL412806)
Affinity DataKd: >501nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077136(CHEMBL3416749)
Affinity DataKd:  135nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077135(CHEMBL3416750)
Affinity DataKd:  31nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077139(CHEMBL3416752)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKd:  509nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd:  353nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075817(CHEMBL2371240 | Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gl...)
Affinity DataKd: >1.00E+5nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075816(CHEMBL264208 | Mca1,D-Trp2,Sar7AVT)
Affinity DataKd:  3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075820(CHEMBL405165 | Mpa-D-Trp-lle-Gln-Asn-Cys-Sar-Arg-G...)
Affinity DataKd:  4.96E+3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075818(CHEMBL157988 | Mpa1,D-Phe2,Sar7AVT)
Affinity DataKd:  421nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397206(CHEMBL2172289)
Affinity DataKd:  1.38nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397207(CHEMBL2172288)
Affinity DataKd:  11.1nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397209(CHEMBL2172291)
Affinity DataKd:  2.53nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397210(CHEMBL2172290)
Affinity DataKd:  2.33nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075817(CHEMBL2371240 | Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gl...)
Affinity DataKd: >1.00E+5nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407332(CHEMBL405005)
Affinity DataKd:  26.9nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407334(CHEMBL1790313)
Affinity DataKd:  3.98E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407336(CHEMBL412616)
Affinity DataKd:  2.88E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407333(CHEMBL412942)
Affinity DataKd:  15.5nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407337(CHEMBL1790314)
Affinity DataKd:  3.16E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407339(CHEMBL1790307)
Affinity DataKd:  3.16E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407335(CHEMBL428187)
Affinity DataKd: >1.26E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407341(CHEMBL264449)
Affinity DataKd:  1.00E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407344(CHEMBL261914)
Affinity DataKd:  1.26E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407343(CHEMBL412806)
Affinity DataKd: >2.51E+3nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407338(CHEMBL385062)
Affinity DataKd:  56.2nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50407349(CHEMBL265357)
Affinity DataKd:  46.8nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50403723(CHEMBL2110163)
Affinity DataKd:  2.29E+3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed