Compile Data Set for Download or QSAR
maximum 50k data
Found 73 of kd data for polymerid = 3929
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM109236(WEHI-539)
Affinity DataIC50: >1.20E+4nM Kd: >550nMpH: 7.4Assay Description:The protocols for tight and weak binders were described in Biacore S51 assay set-up with a flow rate of 30 µL/min. For His-Bcl-2 protein assays...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM218795(130E7 | Ac-λIAQELRRIGDEFNAYYARR-NH2)
Affinity DataKd:  2nMpH: 7.4 T: 2°CAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50020929(CHEMBL3287292)
Affinity DataKd: >2.00E+4nMAssay Description:Binding affinity to Mcl-1 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50020930(CHEMBL3287293)
Affinity DataKd: >2.00E+4nMAssay Description:Binding affinity to Mcl-1 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50020938(CHEMBL3287301)
Affinity DataKd:  1.44E+4nMAssay Description:Binding affinity to Mcl-1 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50041679(CHEMBL3358892)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50041679(CHEMBL3358892)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to human MCL1 (173 to 329 aa) by 19F NMR spectroscopyMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50059666(CHEMBL3393634)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to Mcl1 (unknown origin) assessed as fluorescence quenching by intrinsic fluorescence spectraMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50059667(CHEMBL3393637)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to Mcl1 (unknown origin) assessed as fluorescence quenching by intrinsic fluorescence spectraMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM21400(CHEMBL192571 | N-[(4-{[(2R)-4-(dimethylamino)-1-(p...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to Mcl1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50160008(CHEMBL3785755)
Affinity DataKd:  1.50E+6nMAssay Description:Binding affinity to N-terminal His-tagged human Mcl-1 (172 to 327 residues) expressed in Escherichia coli BL21(DE3) in presence of 6-chloro-3-(3-(4-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50107130((Z)-2-(5-(4-bromobenzylidene)-4-oxo-2-thioxothiazo...)
Affinity DataKd:  4.40E+4nMAssay Description:Displacement of fluorescein-labeled Bak-BH3 peptide from human Mcl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50107130((Z)-2-(5-(4-bromobenzylidene)-4-oxo-2-thioxothiazo...)
Affinity DataKd:  8.40E+4nMAssay Description:Binding affinity to human Mcl1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50308110((S,Z)-2-(5-((6-(2,3-dimethoxyphenyl)pyridin-3-yl)m...)
Affinity DataKd:  6.90E+3nMAssay Description:Displacement of fluorescein-labeled Bak-BH3 peptide from human Mcl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50308110((S,Z)-2-(5-((6-(2,3-dimethoxyphenyl)pyridin-3-yl)m...)
Affinity DataKd:  250nMAssay Description:Binding affinity to human Mcl1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50308111((S,Z)-2-(5-((6-(3,4-dimethoxyphenyl)pyridin-3-yl)m...)
Affinity DataKd:  8.00E+3nMAssay Description:Displacement of fluorescein-labeled Bak-BH3 peptide from human Mcl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50308111((S,Z)-2-(5-((6-(3,4-dimethoxyphenyl)pyridin-3-yl)m...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to human Mcl1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKd:  2.32E+3nMAssay Description:Binding affinity to cMcl-1 (residues 171 to 327) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50424204(CHEMBL2312475)
Affinity DataKd:  802nMAssay Description:Binding affinity to cMcl-1 (residues 171 to 327) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50424209(CHEMBL2312470)
Affinity DataKd:  105nMAssay Description:Binding affinity to cMcl-1 (residues 171 to 327) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50424211(CHEMBL2312484)
Affinity DataKd:  512nMAssay Description:Binding affinity to cMcl-1 (residues 171 to 327) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50336576(3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-...)
Affinity DataKd:  954nMAssay Description:Binding affinity to cMcl-1 (residues 171 to 327) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428724(CHEMBL2333152)
Affinity DataKd:  1.45E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428725(CHEMBL2333151)
Affinity DataKd:  3.71E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428726(CHEMBL2333150)
Affinity DataKd:  4.93E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428727(CHEMBL2333149)
Affinity DataKd:  4.24E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428728(CHEMBL2333148)
Affinity DataKd:  160nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428729(CHEMBL2333147)
Affinity DataKd:  1.58E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428730(CHEMBL2333146)
Affinity DataKd:  4.28E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428731(CHEMBL2333145)
Affinity DataKd:  6.65E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428732(CHEMBL2333144)
Affinity DataKd:  8.27E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428733(CHEMBL2333143)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428734(CHEMBL1927339)
Affinity DataKd:  2.21E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50425963(CHEMBL2314369)
Affinity DataKd:  5.23E+4nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM22853(1,2-Dione-Based Compound, 10 | 1,2-dihydroacenapht...)
Affinity DataKd:  3.25E+5nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428735(CHEMBL2333142 | Cyanoacetamide)
Affinity DataKd:  1.35E+4nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50428736(CHEMBL2333141 | Thiomorpholine)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50345445(8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile |...)
Affinity DataKd:  1.83E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50336576(3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-...)
Affinity DataKd:  960nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKd:  2.65E+3nMAssay Description:Binding affinity to his-tagged Mcl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKd:  2.65E+3nMAssay Description:Binding affinity to Mcl1 (unknown origin) expressed in Escherichia coli BL21 by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50425964(CHEMBL2314383)
Affinity DataKd:  980nMAssay Description:Binding affinity to Mcl1 (unknown origin) expressed in Escherichia coli BL21 by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50336576(3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-...)
Affinity DataKd:  58nMAssay Description:Inhibition of FAM-Bid binding to Mcl-1 (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50303802(CHEMBL4169380)
Affinity DataKd:  150nMAssay Description:Compound was tested for inhibitory activity against Inosine-5'-monophosphate dehydrogenase, the type of inhibition in not competitiveMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50500860(CHEMBL3799447)
Affinity DataKd:  265nMAssay Description:Binding affinity to N-terminal 8x His-tagged MCl-1 (unknown origin) expressed in Escherichia coli BL21 (DE3) by isothermal titration microcalorimetri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM50522905(CHEMBL4593715)
Affinity DataKd:  165nMAssay Description:Binding affinity to biotin-labelled TEV-fused GST-tagged MCl-1 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM203869(7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...)
Affinity DataKd:  0.140nMAssay Description:Binding affinity to MCl-1 (unknown origin) assessed as binding affinity constant for state oneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM203875(7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...)
Affinity DataKd:  0.130nMAssay Description:Binding affinity to MCl-1 (unknown origin) assessed as binding affinity constant for state oneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM203875(7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to MCl-1 (unknown origin) assessed as binding affinity constant for state twoMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

LigandPNGBDBM203869(7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...)
Affinity DataKd:  0.0180nMAssay Description:Binding affinity to MCl-1 (unknown origin) assessed as binding affinity constant for state twoMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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