Found 7 of kd data for polymerid = 50006595 TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Inhibition of 8-NBD-cAMP binding to human EPAC1 cAMP binding domain (149 to 318 residues) by fluorescence assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) using aggregate form of compound by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 1.24E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 4.90E+3nMAssay Description:Binding affinity to GST-tagged human EPAC1 L273W mutant expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by 8-NBD-cAMP based competitiv...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 6.60E+3nMAssay Description:Binding affinity to GST-tagged human EPAC1 CNBD (149 to 318 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by 8-NBD-cAMP ba...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 4.50E+3nMAssay Description:Binding affinity to GST-tagged human EPAC1 CNBD (149 to 318 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by 8-NBD-cAMP ba...More data for this Ligand-Target Pair
3D Structure (crystal)TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 7.57E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) in presence of human serum albumin by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
