Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of kd data for polymerid = 50007553
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50271260(CHEMBL4130196)
Affinity DataKd:  15nMAssay Description:Binding affinity to human GST-tagged TEAD1 (194 to 411) expressed in Escherichia coli BL21(DE3) by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50497296(CHEMBL3335452)
Affinity DataKd:  39nMAssay Description:Inhibition of YAP/ GST-TEAD1 interaction in human Bel-7404 cells by GST pull-down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50497300(CHEMBL3335461)
Affinity DataKd:  15nMAssay Description:Inhibition of YAP/ GST-TEAD1 interaction in human Bel-7404 cells by GST pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  120nMAssay Description:Binding affinity to human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50497304(CHEMBL3335453)
Affinity DataKd:  18nMAssay Description:Inhibition of YAP/ GST-TEAD1 interaction in human Bel-7404 cells by GST pull-down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50531838(Pirazidol | Pirlindole)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to TEAD1 (194 to 411 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50600845(CHEMBL5173440)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity to human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities Of Lille

Curated by ChEMBL
LigandPNGBDBM50497293(CHEMBL3335451)
Affinity DataKd:  211nMAssay Description:Inhibition of YAP/ GST-TEAD1 interaction in human Bel-7404 cells by GST pull-down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed