Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of kd data for polymerid = 6987,7216,50003841
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50126720((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataKd:  3.60nMAssay Description:Equilibrium constant for P2X purinoceptor 7 expressed in HEK 293 cells at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50586608(CHEMBL5083184)
Affinity DataKd:  710nMAssay Description:Binding affinity to human wild type P2X7R assessed as dissociation constant by microscale thermophoresis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50126720((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataKd:  3.60nMAssay Description:Maximum binding affinity towards P2X purinoceptor 7 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed