Compile Data Set for Download or QSAR
maximum 50k data
Found 16 of kd data for polymerid = 7256
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339033(5-[(4-(3S)-4-[(1R,2R)-2-ethoxy-5-(trifluoromethyl)...)
Affinity DataKd:  3.10nMAssay Description:Activation of CCR5 in human PBMC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50509860(CHEMBL4442783)
Affinity DataKd:  24nMAssay Description:Binding affinity to CCR5 in T-cell (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378977(CHEMBL1621896)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378978(CHEMBL2011440)
Affinity DataKd:  1.08E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 after 1 min by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378979(CHEMBL2011441)
Affinity DataKd:  2.86E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 after 1 min by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50334986(4,4-Difluoro-cyclohexanecarboxylic acid {(S)-3-[(1...)
Affinity DataKd:  25nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378980(CHEMBL1618631)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378981(CHEMBL2011439)
Affinity DataKd:  8.20E+3nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378982(CHEMBL1623307)
Affinity DataKd:  2.75E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378983(CHEMBL1907216)
Affinity DataKd:  1.84E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378978(CHEMBL2011440)
Affinity DataKd:  1.75E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378979(CHEMBL2011441)
Affinity DataKd:  2.26E+4nMAssay Description:Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50267124(CHEMBL2163486)
Affinity DataKd:  1.60nMAssay Description:Antagonist activity at human CCR5 expressed in HEK 293 Glosensor cells assessed as reduction in RANTES-induced intracellular calcium levels preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50267125(CHEMBL4089991)
Affinity DataKd:  10nMAssay Description:Antagonist activity at human CCR5 expressed in HEK 293 Glosensor cells assessed as reduction in RANTES-induced intracellular calcium levels preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50267126(CHEMBL4068906)
Affinity DataKd:  316nMAssay Description:Antagonist activity at human CCR5 expressed in HEK 293 Glosensor cells assessed as reduction in RANTES-induced intracellular calcium levels preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336345(4-(4-(((R)-1-butyl-3-((R)-cyclohexyl(hydroxy)methy...)
Affinity DataKd:  3nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed