Compile Data Set for Download or QSAR
maximum 50k data
Found 79 of kd data for polymerid = 866,7224,9862,50000517,50004006,50006580
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000002(CHEMBL2370814 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Lys(a...)
Affinity DataKd:  0.860nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000003(CHEMBL266716 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Arg-(D...)
Affinity DataKd:  0.240nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000005(CHEMBL2370803 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Lys(a...)
Affinity DataKd:  0.860nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000006(CHEMBL2370809 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Lys(N...)
Affinity DataKd:  0.350nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000001(CHEMBL2370818 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Lys(a...)
Affinity DataKd:  0.480nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000004(CHEMBL2370808 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Arg-(...)
Affinity DataKd:  0.670nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50000007(CHEMBL2370807 | [Ac-(D)Nal-(D)Cpa-(D)Pal-Ser-Orn(a...)
Affinity DataKd:  0.210nMAssay Description:The binding affinity towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007944(CHEMBL386314 | pGlu-His-Trp-Ser-NicLys-DNicLys-Leu...)
Affinity DataKd:  0.110nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007945(CHEMBL2369851 | pGlu-His-Trp-Ser-Lys(atz)-DLys(atz...)
Affinity DataKd:  0.480nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007946(CHEMBL428837 | pGlu-His-Trp-Ser-Arg(bCN)-DArg(bCN)...)
Affinity DataKd:  2.10nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007947(CHEMBL269583 | pGlu-His-Trp-Ser-Har(2mpCN)-DHar(2m...)
Affinity DataKd:  0.270nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007948(CHEMBL412802 | pGlu-His-DPal-Ser-Tyr-DHar(bCN)-Leu...)
Affinity DataKd:  1.70nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007949(CHEMBL411586 | pGlu-His-Trp-Ser-Har(bCN)-DHar(bCN)...)
Affinity DataKd:  1.30nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007950(CHEMBL439359 | pGlu-His-Trp-Ser-Har(chCN)-DHar(chC...)
Affinity DataKd:  1.20nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007951(CHEMBL407482 | pGlu-His-DPal-Ser-Tyr-DArg-Leu-Har(...)
Affinity DataKd:  1nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007953(CHEMBL414113 | pGlu-His-DPal-Ser-Tyr-DPal-Leu-ILys...)
Affinity DataKd:  0.0800nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007952(CHEMBL414391 | pGlu-His-Trp-Ser-Har(mCN)-DHar(mCN)...)
Affinity DataKd:  0.240nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007954(CHEMBL407023 | pGlu-His-DHar(bCN)-Ser-Tyr-DArg-Leu...)
Affinity DataKd:  1.20nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007957(CHEMBL438191 | pGlu-His-Trp-Ser-NicLys-DNicLys-Leu...)
Affinity DataKd:  0.450nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007955(CHEMBL218396 | pGlu-His-DLys(atz)-Ser-Tyr-DArg-Leu...)
Affinity DataKd:  0.270nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007956(CHEMBL265522 | pGlu-His-Trp-Ser-Har(hCN)-DHar(hCN)...)
Affinity DataKd:  3.30nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007959(CHEMBL438762 | pGlu-His-Trp-Ser-Har(iCN)-DHar(iCN)...)
Affinity DataKd:  0.320nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007958(CHEMBL2369860 | pGlu-His-Trp-Ser-Orn(atz)-DOrn(atz...)
Affinity DataKd:  0.210nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50007960(CHEMBL261999 | pGlu-His-Trp-Ser-Arg(2mpCN)-DArg(2m...)
Affinity DataKd:  0.410nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataKd:  375nMAssay Description:Binding affinity at Leutinizing releasing hormone receptor in rat pituitary using [125I]-leuprolide as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataKd:  811nMAssay Description:In vitro inhibition of Escherichia coli dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataKd:  221nMAssay Description:In vitro inhibition of dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022922(Ac-DNal-DCpa-DPal-c[Dpr-Arg-DPal-Leu-Arg-Pro-Asp]-...)
Affinity DataKd:  4.5nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022912(Ac-DNal-DCpa-DPal-c[Cys-Arg-DPal-Leu-Arg-Pro-Cys]-...)
Affinity DataKd:  0.800nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022913(Ac-DNal-DFpa-DTrp-Ser-Tyr-DArg-Leu-Arg-Pro-Gly-NH2...)
Affinity DataKd:  0.640nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022914(Ac-DNal-DFpa-DTrp-[Dpr-Tyr-DArg-Leu-Arg-Pro-Asp]-N...)
Affinity DataKd:  1.90nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022916(Ac-delta3-Pro-DFpa-DTrp-Ser-Tyr-DTrp-Leu-Arg-Pro-G...)
Affinity DataKd:  0.270nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022917(Ac-DNal-DFpa-DTrp-[Cys-Tyr-DArg-Leu-Arg-Pro-Cys]-N...)
Affinity DataKd:  6nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022918(Ac-DNal-DCpa-DPal-Ser-Arg-DPal-Leu-Arg-Pro-DAla-NH...)
Affinity DataKd:  0.240nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022915(Ala-Phe-Trp-Ser-Tyr-Arg-Leu-Arg-Asp-Gly | CHEMBL26...)
Affinity DataKd: >100nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022919(Ac-DNal-DFpa-DTrp-[Asp-Tyr-DArg-Leu-Arg-Pro-Dpr]-N...)
Affinity DataKd:  10nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022920(Ac-DNal-DCpa-DPal-c[Glu-Arg-DPal-Leu-Arg-Pro-Dpr]-...)
Affinity DataKd:  1nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022921(Ac-DNal-DCpa-DPal-c[Asp-Arg-DPal-Leu-Arg-Pro-Orn]-...)
Affinity DataKd:  11nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022923(Ac-DNal-DFpa-DTrp-[Glu-Tyr-DArg-Leu-Arg-Pro-Dpr]-N...)
Affinity DataKd:  1.10nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022924(Ac-DNal-DCpa-DPal-Dpr(Ac)-Arg-DPal-Leu-Arg-Pro-Asn...)
Affinity DataKd:  1nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022925(Ac-DNal-DFpa-DTrp-[Asp-Tyr-DArg-Leu-Arg-Pro-Orn]-N...)
Affinity DataKd:  41nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50022926(Ac-DNal-DCpa-DPal-c[Asp-Arg-DPal-Leu-Arg-Pro-Dpr]-...)
Affinity DataKd:  1.10nMAssay Description:Inhibitory binding constant for Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102453(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Hor)]-D-[Amf(...)
Affinity DataKd:  0.794nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102454(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-Tyr-D-Har(Et2)-Leu...)
Affinity DataKd:  0.501nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102467(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Hor)]-D-[Aph(...)
Affinity DataKd:  1nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102459(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(DHor)]-D-[Amf...)
Affinity DataKd:  1.58nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102443(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Cbm)]-D-[Aph(...)
Affinity DataKd:  1.58nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102444(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Hor)]-D-[Amf(...)
Affinity DataKd:  1nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50209591(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Atz)]-D-[Aph(...)
Affinity DataKd:  1.58nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102441(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Hor)]-D-[Amf(...)
Affinity DataKd:  1.26nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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