Affinity DataKi: 0.0220nMAssay Description:Inhibitory activity against adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0628nMAssay Description:Displacement of [3H]DPCPX from rat adenosine receptor A1 by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0709nMAssay Description:Displacement of [3H]DPCPX from rat adenosine receptor A1 by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0867nMAssay Description:Displacement of [3H]DPCPX from rat adenosine receptor A1 by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0940nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]- CHA or [3H]- PIA in bovine brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.124nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortex membranes incubated for 90 mins by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.124nMAssay Description:Binding affinity to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.155nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.155nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.175nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Sprague-Dawley rat whole brain after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:In vitro binding affinity for Adenosine A1 receptor of bovine cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.183nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity towards adenosine A1 receptor in rat forebrain membranes using N6-[3H]cyclohexyladenosineMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity at bovine Adenosine A1 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortical membrane in presence of 100 uM GTPMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortex membranes incubated for 90 mins by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.211nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in presence of 0.1 mM GTPMore data for this Ligand-Target Pair
Affinity DataKi: 0.216nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity for Adenosine A1 receptor using [3H]- CHA or [3H]- PIAMore data for this Ligand-Target Pair
Affinity DataKi: 0.229nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Inhibition of N6-[3H]cyclohexyladenosine binding to adenosine A1 receptor from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity against Adenosine A1 receptor from rat forebrain membranes with N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]-cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
Affinity DataKi: 0.237nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity against Adenosine A1 receptor using [3H]CHA in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to bovine brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Adenosine A1 receptor binding using [3H]DPCPX in rat cortical membranesMore data for this Ligand-Target Pair