Compile Data Set for Download or QSAR
Report error Found 5 of koff data for polymerid = 236,1043,1045,1064,3619,3621,4933,50000072,50006985,50007874,236,1043,1045,1064,3619
TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50093799((R)-1-Amino-13-ethylidene-8,8,11-trimethyl-6-aza-t...)
Affinity DataKon:  0.000217M-1s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKon:  0.000333M-1s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKon:  0.000367M-1s-1 Koff:  0.0155s-1Assay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
In DepthDetails Article

TargetAcetylcholinesterase(Pacific electric ray)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50138279(CHEMBL3752467)
Affinity DataKon:  0.0310M-1s-1Assay Description:Noncompetitive inhibition of Torpedo californica AChE using ATCh as substrate assessed as dissociation rate constant preincubated for 90 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Pacific electric ray)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50138279(CHEMBL3752467)
Affinity DataKon:  0.0320M-1s-1Assay Description:Competitive inhibition of Torpedo californica AChE using ATCh as substrate assessed as dissociation rate constant preincubated for 90 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)