Compile Data Set for Download or QSAR
Report error Found 83 of kon data for polymerid = 236,1043,1045,1064,3619,3621,4933,50000072,50006985,50007874,236,1043,1045,1064,3619
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064504BDBM50064504(CHEMBL3401226)
Affinity DataKoff:  433s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064503BDBM50064503(CHEMBL3401225)
Affinity DataKoff:  6.32E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064502BDBM50064502(CHEMBL3401224)
Affinity DataKoff:  3.00E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064501BDBM50064501(CHEMBL3401223)
Affinity DataKoff:  1.80E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064499BDBM50064499(CHEMBL3401222)
Affinity DataKoff:  3.10E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016939BDBM50016939(CHEMBL3277096)
Affinity DataKoff:  2.50E+4s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064496BDBM50064496(CHEMBL3401221)
Affinity DataKoff:  1.53E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016940BDBM50016940(Ecothiopate Iodide | Phospholine Iodide | CHEBI:59...)
Affinity DataKoff:  4.33E+4s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064493BDBM50064493(CHEMBL3401220)
Affinity DataKoff:  1.24E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064492BDBM50064492(CHEMBL3401219)
Affinity DataKoff:  2.40E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016935BDBM50016935(CHEMBL3277092)
Affinity DataKoff:  68.3s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016936BDBM50016936(CHEMBL3277093)
Affinity DataKoff:  18.3s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064491BDBM50064491(CHEMBL3401218)
Affinity DataKoff:  1.35E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016937BDBM50016937(CHEMBL3277094)
Affinity DataKoff:  0.430s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064490BDBM50064490(CHEMBL3401217)
Affinity DataKoff:  437s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016938BDBM50016938(CHEMBL3277095)
Affinity DataKoff:  13.3s-1Assay Description:Inhibition of electric eel AChE assessed as decrease in thiophenol formation using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064489BDBM50064489(CHEMBL3401216)
Affinity DataKoff:  1.87E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064488BDBM50064488(CHEMBL3401215)
Affinity DataKoff:  515s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064487BDBM50064487(CHEMBL3401214)
Affinity DataKoff:  3.32E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064486BDBM50064486(CHEMBL3401213)
Affinity DataKoff:  5.18E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064485BDBM50064485(CHEMBL3401212)
Affinity DataKoff:  1.13E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064484BDBM50064484(CHEMBL3401211)
Affinity DataKoff:  3.62E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Bovine)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027343BDBM50027343(CHEBI:75701 | ISOPROPYL METHYLPHOSPHONOFLUORIDATE)
Affinity DataKoff:  1.23E+4s-1Assay Description:Inhibition of bovine AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064483BDBM50064483(CHEMBL3401210)
Affinity DataKoff:  3.88E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064481BDBM50064481(CHEMBL3401209)
Affinity DataKoff:  9.35E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Bovine)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027342BDBM50027342(CHEMBL483105)
Affinity DataKoff:  1.10E+5s-1Assay Description:Inhibition of bovine AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064480BDBM50064480(CHEMBL3401208)
Affinity DataKoff:  1.72E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064479BDBM50064479(CHEMBL3401207)
Affinity DataKoff:  20.3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064478BDBM50064478(ALDICARB)
Affinity DataKoff:  108s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064477BDBM50064477(CHEMBL3401206)
Affinity DataKoff:  1.34E+4s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027341BDBM50027341(CHEBI:38721 | METHAMIDOPHOS)
Affinity DataKoff:  32s-1Assay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064476BDBM50064476(CHEMBL2046821 | 3-Tert-Butylphenyl Methylcarbamate)
Affinity DataKoff:  2.10E+3s-1Assay Description:Inhibition of recombinant human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10620BDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataKoff:  55s-1Assay Description:Inhibition of human AChE assessed as carbamylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027343BDBM50027343(CHEBI:75701 | ISOPROPYL METHYLPHOSPHONOFLUORIDATE)
Affinity DataKoff:  4.50E+5s-1Assay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10620BDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataKoff:  0.0333s-1Assay Description:Inhibition of Torpedo californica AChE assessed as carbamylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027342BDBM50027342(CHEMBL483105)
Affinity DataKoff:  2.00E+6s-1Assay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027340BDBM50027340(FENAMIPHOS)
Affinity DataKoff:  0.330s-1Assay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50022772BDBM50022772(Isopropyl phosphorofluoridate | Neoglaucit | O,O'-...)
Affinity DataKoff:  2.17E+3s-1Assay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
University of Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10620BDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataKoff:  0.0333s-1Assay Description:Pseudo-irreversible inhibition of Torpedo californica AChE using acetylthiocholine as substrate by cornish bowden plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490822BDBM50490822(2-Fluoroethyl 4-Nitrophenyl Methylphosphonate | CH...)
Affinity DataKoff:  233s-1Assay Description:Inhibition of human recombinant AChE by time-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490821BDBM50490821(2-Fluoroethyl 4-Nitrophenyl Ethylphosphonate | CHE...)
Affinity DataKoff:  1.03E+3s-1Assay Description:Inhibition of human recombinant AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490822BDBM50490822(2-Fluoroethyl 4-Nitrophenyl Methylphosphonate | CH...)
Affinity DataKoff:  983s-1Assay Description:Inhibition of electric eel AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
The University of Montana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490822BDBM50490822(2-Fluoroethyl 4-Nitrophenyl Methylphosphonate | CH...)
Affinity DataKoff:  1.02E+3s-1Assay Description:Inhibition of rat brain AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
The University of Montana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240416BDBM50240416(diethyl 4-nitrophenyl phosphate | paraoxon | O,O-d...)
Affinity DataKoff:  267s-1Assay Description:Inhibition of rat brain AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Virginia Tech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490822BDBM50490822(2-Fluoroethyl 4-Nitrophenyl Methylphosphonate | CH...)
Affinity DataKoff:  1.25E+3s-1Assay Description:Inhibition of human recombinant AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240416BDBM50240416(diethyl 4-nitrophenyl phosphate | paraoxon | O,O-d...)
Affinity DataKoff:  333s-1Assay Description:Inhibition of electric eel AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490824BDBM50490824(CHEMBL2348369)
Affinity DataKoff:  200s-1Assay Description:Inhibition of electric eel AChE by time-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
The University of Montana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240416BDBM50240416(diethyl 4-nitrophenyl phosphate | paraoxon | O,O-d...)
Affinity DataKoff:  567s-1Assay Description:Inhibition of rat brain AChE by time-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490821BDBM50490821(2-Fluoroethyl 4-Nitrophenyl Ethylphosphonate | CHE...)
Affinity DataKoff:  917s-1Assay Description:Inhibition of electric eel AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
The University of Montana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490821BDBM50490821(2-Fluoroethyl 4-Nitrophenyl Ethylphosphonate | CHE...)
Affinity DataKoff:  200s-1Assay Description:Inhibition of rat brain AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
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