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Report error Found 4 Enz. Inhib. hit(s) for PDB: 1UK0
TargetPoly [ADP-ribose] polymerase 1(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM27709(2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Bovine)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM27709(2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50:  16nMAssay Description:Inhibition of calf thymus PARP-1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM27709(2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant PARP1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM27709(2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50:  16nMpH: 8.0 T: 23°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair