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Report error Found 3 Enz. Inhib. hit(s) for PDB: 3B28
TargetHeat shock protein HSP 90-alpha(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50354813(CHEMBL1834096)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged HSP90alpha expressed in Escherichia coli after 1 hr using 10 mM of ATP and malachite green by microplate re...Checked by AuthorMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50354813(CHEMBL1834096)
Affinity DataKd:  3.40nMAssay Description:Binding affinity towards N-terminal biotinylated human HSP90-alpha (9 to 236 residues) measured by surface plasmon resonance (SPR) assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50354813(CHEMBL1834096)
Affinity DataKd:  3.40nMAssay Description:Binding affinity to human HSP90alpha assessed as 2D1H-15N chemical shift perturbation by NMR spectroscopyChecked by AuthorMore data for this Ligand-Target Pair