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Report error Found 2 Enz. Inhib. hit(s) for PDB: 4PVU
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266372(CHEMBL451321 | metaglidasen)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266372(CHEMBL451321 | metaglidasen)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galac...More data for this Ligand-Target Pair