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Report error Found 2 Enz. Inhib. hit(s) for PDB: 6MXZ
TargetTP53-binding protein 1(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM154564(N-(3-(Tert-butylamino)propyl)-3-isopropylbenzamide...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of 53BP1 methyllysine binding domain (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTP53-binding protein 1(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM154564(N-(3-(Tert-butylamino)propyl)-3-isopropylbenzamide...)
Affinity DataIC50:  1.40E+4nMpH: 8.0 T: 1,117.6°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)