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Found 5 Enz. Inhib. hit(s) with Target = 'Colony stimulating factor 1 receptor'
TargetColony stimulating factor 1 receptor(Canis lupus familiaris (Dog) (Canis familiaris))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM276744(US10071991, Compound (I-M2-2S,4R) | US10800764, Co...)
Affinity DataIC50:  2nMpH: 7.0 T: 2°CAssay Description:In this assay, recombinant human, dog or rat c-fms catalyzed the phosphorylation of the FMS peptide substrate, SYEGNSYTFIDPTQ, with the phosphorylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetColony stimulating factor 1 receptor(Canis lupus familiaris (Dog) (Canis familiaris))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM276745(US10071991, Compound (I-M2-2R,4S) | US10800764, Co...)
Affinity DataIC50:  2nMpH: 7.0 T: 2°CAssay Description:In this assay, recombinant human, dog or rat c-fms catalyzed the phosphorylation of the FMS peptide substrate, SYEGNSYTFIDPTQ, with the phosphorylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetColony stimulating factor 1 receptor(Canis lupus familiaris (Dog) (Canis familiaris))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM276746(US10071991, Compound (I-M7-2S,4R) | US11214566, Co...)
Affinity DataIC50:  6.60nMpH: 7.0 T: 2°CAssay Description:In this assay, recombinant human, dog or rat c-fms catalyzed the phosphorylation of the FMS peptide substrate, SYEGNSYTFIDPTQ, with the phosphorylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetColony stimulating factor 1 receptor(Canis lupus familiaris (Dog) (Canis familiaris))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM276747(US10071991, Compound (I-M7-2R,4S))
Affinity DataIC50:  8nMpH: 7.0 T: 2°CAssay Description:In this assay, recombinant human, dog or rat c-fms catalyzed the phosphorylation of the FMS peptide substrate, SYEGNSYTFIDPTQ, with the phosphorylate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetColony stimulating factor 1 receptor(Canis lupus familiaris (Dog) (Canis familiaris))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM276743(US10071991, Compound (P) | US10800764, Compound (P...)
Affinity DataIC50:  16nMpH: 7.0 T: 2°CAssay Description:In this assay, recombinant human, dog or rat c-fms catalyzed the phosphorylation of the FMS peptide substrate, SYEGNSYTFIDPTQ, with the phosphorylate...More data for this Ligand-Target Pair
In DepthDetails US Patent