Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [G719S]'
TargetEpidermal growth factor receptor [G719S](Homo sapiens (Human))
Synovo

US Patent
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  6.70nMpH: 7.5 T: 2°CAssay Description:FlashPlates from Perkin Elmer (Boston, Mass., USA) with a 50 μl reaction volume are used. The reaction cocktail was pipetted in 4 steps in the fol...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [G719S](Homo sapiens (Human))
Synovo

US Patent
LigandPNGBDBM50379214(CHEMBL2011291 | US9416123, 6)
Affinity DataIC50:  2.60E+3nMpH: 7.5 T: 2°CAssay Description:FlashPlates from Perkin Elmer (Boston, Mass., USA) with a 50 μl reaction volume are used. The reaction cocktail was pipetted in 4 steps in the fol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor [G719S](Homo sapiens (Human))
Synovo

US Patent
LigandPNGBDBM373711(US10246444, Example 40)
Affinity DataKd:  50nMAssay Description:KINOMEscan is based on a competition binding assay that quantitatively measures the ability of a compound to compete with an immobilized, active-site...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent