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Found 8 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase PRDM9 [195-385]'
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228646(H3 (1-25) K4me0 | MARTKQTARKSTGGKAPRKQLATKA)
Affinity DataKd:  3.60E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228647(H3 (1-25) K4me1 | MARTKQTARKSTGGKAPRKQLATKA)
Affinity DataKd:  4.70E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228648(H3 (1-25) K4me2 | MARTKQTARKSTGGKAPRKQLATKA)
Affinity DataKd:  5.80E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228653(H3 (21-44) K36me3 | LATKAARKSAPSTGGVKKPHRYRP)
Affinity DataKd:  9.60E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228650(H3 (21-44) K36me0 | LATKAARKSAPSTGGVKKPHRYRP)
Affinity DataKd:  4.60E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228651(H3 (21-44) K36me1 | LATKAARKSAPSTGGVKKPHRYRP)
Affinity DataKd:  4.10E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228652(H3 (21-44) K36me2 | LATKAARKSAPSTGGVKKPHRYRP)
Affinity DataKd:  4.20E+3nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase PRDM9 [195-385](Homo sapiens (Human))
University Of Toronto

LigandPNGBDBM228649(H3 (1-25) K4me3 | MARTKQTARKSTGGKAPRKQLATKA)
Affinity DataKd:  1.20E+4nMpH: 8.5 T: 2°CAssay Description:In this assay [3H]AdoMet (PerkinElmer Life Sciences; catalog number NET155V250UC)was used as a methyl donor to methylate biotinylated histone peptide...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed