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Found 42 Enz. Inhib. hit(s) with Target = 'Isoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)'
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204852(US9242977, 85-226)
Affinity DataIC50:  1nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204849(US9242977, 85-184)
Affinity DataIC50:  2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204842(US9242977, 71)
Affinity DataIC50:  2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204848(US9242977, 85-117)
Affinity DataIC50:  2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204837(US9242977, 65-1)
Affinity DataIC50:  2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204835(US9242977, 57)
Affinity DataIC50:  3nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204851(US9242977, 85-225)
Affinity DataIC50:  4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204830(US9242977, 23)
Affinity DataIC50:  4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204838(US9242977, 66-19)
Affinity DataIC50:  4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204850(US9242977, 85-209)
Affinity DataIC50:  4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204834(US9242977, 54)
Affinity DataIC50:  4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50:  6nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204832(US9242977, 48)
Affinity DataIC50:  10nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204839(US9242977, 66-27)
Affinity DataIC50:  10nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204843(US9242977, 72-1)
Affinity DataIC50:  11nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204833(US9242977, 50)
Affinity DataIC50:  12nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204840(US9242977, 66-28)
Affinity DataIC50:  14nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204844(US9242977, 72-3)
Affinity DataIC50:  18nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204848(US9242977, 85-117)
Affinity DataIC50:  20nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204838(US9242977, 66-19)
Affinity DataIC50:  20nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204842(US9242977, 71)
Affinity DataIC50:  30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204835(US9242977, 57)
Affinity DataIC50:  30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204845(US9242977, 72-7)
Affinity DataIC50:  30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204841(US9242977, 66-72)
Affinity DataIC50:  32nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204845(US9242977, 72-7)
Affinity DataIC50:  33nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204834(US9242977, 54)
Affinity DataIC50:  40nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204833(US9242977, 50)
Affinity DataIC50:  40nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204841(US9242977, 66-72)
Affinity DataIC50:  50nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204843(US9242977, 72-1)
Affinity DataIC50:  50nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204844(US9242977, 72-3)
Affinity DataIC50:  60nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204836(US9242977, 59)
Affinity DataIC50:  70nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204846(US9242977, 80-2)
Affinity DataIC50:  70nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204840(US9242977, 66-28)
Affinity DataIC50:  80nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204837(US9242977, 65-1)
Affinity DataIC50:  80nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204847(US9242977, 84-41)
Affinity DataIC50:  90nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204830(US9242977, 23)
Affinity DataIC50:  90nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204829(US9242977, 9)
Affinity DataIC50:  93nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204832(US9242977, 48)
Affinity DataIC50:  120nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204839(US9242977, 66-27)
Affinity DataIC50:  130nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204829(US9242977, 9)
Affinity DataIC50:  160nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50:  180nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM204836(US9242977, 59)
Affinity DataIC50:  190nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent