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Found 957 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase'
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50108119(CHEMBL3600587)
Affinity DataKi:  1nMAssay Description:Reversible inhibition of STS (unknown origin) using 4-MUS as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50108118(CHEMBL3600594)
Affinity DataKi:  2.5nMAssay Description:Reversible inhibition of STS (unknown origin) using 4-MUS as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50161121(4-(4-Bromo-2,5-dichloro-thiophene-3-sulfonylaminoc...)
Affinity DataKi:  12nMAssay Description:Inhibitory constant against human Steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50363580(CHEMBL1945908)
Affinity DataKi:  23nMAssay Description:Inhibition of steroid sulfatase using 4-methylumbelliferyl sulfate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  30nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134333(CHEMBL331089 | Phenyl-acetic acid (1R,3R,5S)-8-(3,...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity against Steroid sulfatase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134333(CHEMBL331089 | Phenyl-acetic acid (1R,3R,5S)-8-(3,...)
Affinity DataKi:  76nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  85nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  90nMAssay Description:Mixed type inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50363580(CHEMBL1945908)
Affinity DataKi:  108nMAssay Description:Mixed type inhibition of steroid sulfatase using 4-methylumbelliferyl sulfate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50135162(CHEMBL147705 | Sulfamic acid 2-adamantan-1-yl-4-ox...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50118560(CHEMBL262050 | Sulfamic acid 2-adamantan-1-yl-4-ox...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50161124(4-(3,5-Bis-trifluoromethyl-benzenesulfonylaminocar...)
Affinity DataKi:  220nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355372(CHEMBL482212)
Affinity DataKi:  250nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50168215(CHEMBL3804916)
Affinity DataKi:  250nMAssay Description:Reversible inhibition of human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50525262(CHEMBL4444347)
Affinity DataKi:  350nMAssay Description:Inhibition of sulfatase (unknown origin) using [3H]E1S as substrate after 20 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50112876(3-((N-cyclohexyl-aminocarbonoyl)hydrazono]methyl)-...)
Affinity DataKi:  350nMAssay Description:Non-competitive inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 20 mins by Lineweaver-Burk plot a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  470nMAssay Description:Inhibitory constant against human steroid sulfatase in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151137(2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxyli...)
Affinity DataKi:  500nMAssay Description:Reversible inhibition of recombinant human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151142(2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic ac...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134332(CHEMBL332811 | Phenyl-acetic acid (1R,3R,5S)-8-(4-...)
Affinity DataKi:  530nMAssay Description:Inhibitory constant against purified human Steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151137(2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxyli...)
Affinity DataKi:  530nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  670nMAssay Description:Inhibitory activity against purified human Steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  670nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  670nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134335(8-[N-(4-chlorophenylsulfonamido)-carbonyl amino]-8...)
Affinity DataKi:  890nMAssay Description:Inhibitory activity against Steroid sulfatase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50168258(CHEMBL3805369)
Affinity DataKi:  890nMAssay Description:Inhibition of recombinant human estrone sulfatase expressed in CHO cells using 4-methylumbelliferyl sulfate as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355361(CHEMBL1835541)
Affinity DataKi:  1.40E+3nMAssay Description:Non-Competitive inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Reversible inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134325(CHEMBL440159 | Phenyl-acetic acid (1R,3R,5S)-8-(4-...)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibitory activity against Steroid sulfatase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151135((2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-oxo-aceti...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134328(CHEMBL124349 | Phenyl-acetic acid (1R,3R,5S)-8-(4-...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against Steroid sulfatase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134328(CHEMBL124349 | Phenyl-acetic acid (1R,3R,5S)-8-(4-...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50168216(CHEMBL3806006)
Affinity DataKi:  2.80E+3nMAssay Description:Reversible inhibition of human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151140(2-Adamantan-1-yl-6-(2-hydroxy-acetyl)-chromen-4-on...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134337(CHEMBL121068 | Phenyl-acetic acid (1R,3R,5S)-8-(4-...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibitory constant against purified human Steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibitory constant against human steroid sulfatase in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50161118(4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperazi...)
Affinity DataKi:  1.45E+4nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366322(CHEMBL2367489)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity against estrone sulfatase in placental preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50223216(CHEMBL3348562)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibitory activity against steroid sulfatase (STS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50161119(4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperidi...)
Affinity DataKi:  1.61E+4nMAssay Description:Inhibitory constant against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151134(2-Adamantan-1-yl-4-oxo-4H-chromene-6-carbaldehyde ...)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50370691(CHEMBL1628004)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of sulfatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50370691(CHEMBL1628004)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 8.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50151141(2-Adamantan-1-yl-6-hydroxymethyl-chromen-4-one | C...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366322(CHEMBL2367489)
Affinity DataKi:  3.30E+4nMAssay Description:Binding affinity against estrone sulfatase in breast tumor preparationsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50073853(CHEMBL33862 | Sulfamic acid 4-{(E)-1-[4-(2-dimethy...)
Affinity DataKi:  3.59E+4nMAssay Description:Inhibition of sulfatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Rattus norvegicus)
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50073853(CHEMBL33862 | Sulfamic acid 4-{(E)-1-[4-(2-dimethy...)
Affinity DataKi:  3.59E+4nMAssay Description:In vitro binding affinity against estrone sulfatase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366887(CHEMBL1627329)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibitory activity against steroid sulfatase (STS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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