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Found 45 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein phosphatase non-receptor type 13'
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM199180(US9217012, 10)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 7.0 T: 2°CAssay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in DMG buffer (50 mM DMG, pH 7.0, 1 mM EDTA, 150 mM NaCl, 2 mM DTT, 0.1 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50436358(CHEMBL2396718)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant FAP-1 (unknown origin) using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099713(CHEMBL50878 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50:  600nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50425807(CHEMBL2316902)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50425806(CHEMBL2316907)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50425808(CHEMBL2316906)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50436357(CHEMBL2396719)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of recombinant FAP-1 (unknown origin) using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM84581(Thioxothiazolidinone derivative, 1)
Affinity DataIC50:  3.70E+3nMpH: 7.0 T: 2°CAssay Description:PTP assay were conducted at 25 C in 96-well plates. Reaction rates were determined using a Variokan plate reader from Thermo Electron. For assay pH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099746(CHEMBL51579 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099737(2-Amino-phenanthrene-9,10-dione | CHEMBL417727 | U...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory concentration against FAP-1 using pNPP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099692(CHEMBL51314 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099697(7-(9,10-Dioxo-9,10-dihydro-phenanthren-2-ylcarbamo...)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50607111(CHEMBL5218807)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FAP-1(unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM231167(US9340574, 7)
Affinity DataIC50: >1.00E+4nMpH: 7.0Assay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in 3,3-dimethylglutarate buffer (50 mM 3,3-dimethylglutarate, pH 7.0, 1 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099700(CHEMBL51776 | N-[7-(3-Methoxycarbonyl-propionylami...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099710(Benzo[h]quinoline-5,6-dione | CHEMBL50627)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099717(CHEMBL300241 | [(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory concentration against FAP-1 pNPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099713(CHEMBL50878 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50308158(3-(1-(3-(Biphenyl-4-ylamino)-3-oxopropyl)-1H-1,2,3...)
Affinity DataIC50:  2.03E+4nMpH: 7.0Assay Description:Inhibition of FAP1 expressed in Escherichia coli assessed as inhibition of p-nitrophenyl phosphate hydrolysis at pH 7 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099700(CHEMBL51776 | N-[7-(3-Methoxycarbonyl-propionylami...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099692(CHEMBL51314 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099692(CHEMBL51314 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of protein tyrosine phosphatase N13 (unknown origin) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099697(7-(9,10-Dioxo-9,10-dihydro-phenanthren-2-ylcarbamo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099737(2-Amino-phenanthrene-9,10-dione | CHEMBL417727 | U...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099717(CHEMBL300241 | [(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099710(Benzo[h]quinoline-5,6-dione | CHEMBL50627)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50099746(CHEMBL51579 | N-(9,10-Dioxo-9,10-dihydro-phenanthr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration against FAP-1 using lck-10 mer as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50544440(CHEMBL4647367 | US11192850, Entry 4t)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50544431(CHEMBL4637459 | US11192850, Entry 4k)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558482(CHEMBL4742123)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50335895(6-hydroxy-3-(1-(4-(naphthalen-1-ylamino)-4-oxobuty...)
Affinity DataIC50:  3.68E+4nMAssay Description:Inhibition of FAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50343148(CHEMBL1773181 | N1-(1-(4-(4-fluorophenyl)piperazin...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human FAP1 expressed in Escherichia coli after 5 mins by microplate spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50544427(CHEMBL4632818 | US11192850, Entry 4g)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FAP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50343142(CHEMBL1773168 | N-(4-butylphenyl)-2-oxo-1,2-dihydr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human FAP1 expressed in Escherichia coli after 5 mins by microplate spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50343147(CHEMBL1773180 | N1-(furan-2-ylmethyl)-N2-(1-(4-(4-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human FAP1 expressed in Escherichia coli after 5 mins by microplate spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558487(CHEMBL4786243)
Affinity DataIC50:  7.35E+4nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558481(CHEMBL4783639)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558461(CHEMBL4760367)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558485(CHEMBL4800195)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50607110(CHEMBL5219519)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of FAP-1(unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558488(CHEMBL4794972)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of FAP-1(unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558484(CHEMBL4748824)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558483(CHEMBL4778085)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558488(CHEMBL4794972)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 13(Homo sapiens (Human))
Indiana University Research And Technology

US Patent
LigandPNGBDBM50558486(CHEMBL4797766)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged FAP1 (unknown origin) expressed in Escherichia coli BL21 cells using para-nitrophenyl phosphate as substrate incubated for 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed