Report error Found 3502 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A'
Affinity DataKd: 1.30E+4nMAssay Description:Binding affinity to 5HT3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 7.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Binding affinity against human 5-hydroxytryptamine 3A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in xenopus oocytes by electrophysiological methodMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human 5-HT3 receptor by FLIPR/summary (Abse5) assayMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human 5-HT3 receptor by FLIPR(Abse5) assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.60nMAssay Description:Compound was tested in vitro for its antagonistic activity against 5-hydroxytryptamine 3 receptor in rat CNS.More data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Compound was tested for its antagonistic activity against 5-hydroxytryptamine 3 receptor in rat brain using [3H]zacopride as the radioligand.More data for this Ligand-Target Pair
Affinity DataKd: 0.150nMAssay Description:Compound was tested for its binding affinity towards 5-hydroxytryptamine 3 receptor in whole rat brain using (S)-[125I]-zacopride as the radioligand.More data for this Ligand-Target Pair
Affinity DataEC50: 141nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Affinity DataEC50: 9.20nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 14.5nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 12.6nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at human recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Antagonist activity at rat recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Response at rat 5-hydroxytryptamine 3a receptor expressed in xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 457nMAssay Description:Antagonist activity at human 5HT3A receptor expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at human wild type 5-HT3A/5-HT3B receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at human wild type 5-HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Binding affinity to human wild type 5-HT3A/5-HT3B receptor expressed in HEK293 cells after 24 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Binding affinity to human wild type 5-HT3A receptor expressed in HEK293 cells after 24 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
