Compile Data Set for Download or QSAR
Report error Found 14020 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1'
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21222(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21223(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21224(N-[2-(methylsulfanyl)-6-propoxypyrimidin-4-yl]acet...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21225(N-[2-(methylsulfanyl)-6-propoxypyrimidin-4-yl]prop...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21226(N-[6-methoxy-2-(propylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21230(N-[2-(benzylsulfanyl)-6-propoxypyrimidin-4-yl]acet...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21234(N-{6-[(4-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21235(N-{6-[(2,4-dichlorophenyl)methoxy]-2-(propylsulfan...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21238(N-[6-(cyclohexylmethoxy)-2-(propylsulfanyl)pyrimid...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21240(N-[2-(tert-butylsulfanyl)-6-[(4-chlorophenyl)metho...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM198127(4-amino-6-alkyloxy-2-benzylthiopyrimidines (4))
Affinity DataEC50:  490nMpH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM198128(4-amino-6-alkyloxy-2-benzylthiopyrimidines (5))
Affinity DataEC50:  870nMpH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKd:  3nMpH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191774(US9187428, 2)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191775(US9187428, 3)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191776(US9187428, 53 | US9187428, 4)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191778(US9187428, 6)
Affinity DataEC50:  0.0600nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191779(US9187428, 7)
Affinity DataEC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191785(US9187428, 13)
Affinity DataEC50:  0.0800nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191786(US9187428, 14)
Affinity DataEC50:  3.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191787(US9187428, 15)
Affinity DataEC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191793(US9187428, 21)
Affinity DataEC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191798(US9187428, 26)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191799(US9187428, 27)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191800(US9187428, 28)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191801(US9187428, 29)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191802(US9187428, 30)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191803(US9187428, 31)
Affinity DataEC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191804(US9187428, 32)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191805(US9187428, 33)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191809(US9187428, 37)
Affinity DataEC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191810(US9187428, 38)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191816(US9187428, 44)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191818(US9187428, 46)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191821(US9187428, 49)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191822(US9187428, 50)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191823(US9187428, 51)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191776(US9187428, 53 | US9187428, 4)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191826(US9187428, 54)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191827(US9187428, 55)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
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US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191828(US9187428, 56)
Affinity DataEC50:  2.80nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191832(US9187428, 60)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191834(US9187428, 62)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191837(US9187428, 65)
Affinity DataEC50:  3.30nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191838(US9187428, 66)
Affinity DataEC50:  1.30nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191840(US9187428, 68)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191842(US9187428, 70)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191844(US9187428, 72)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191846(US9187428, 74)
Affinity DataEC50:  2.40nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Human)
Universita Di Napoli

LigandPNGBDBM191847(US9187428, 75)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent

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