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Report error Found 42 Enz. Inhib. hit(s) with Target = 'CTP synthase 1'
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609673(CHEMBL5267968)
Affinity DataIC50:  13nMAssay Description:Inhibition of human CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Mus musculus)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609673(CHEMBL5267968)
Affinity DataIC50:  18nMAssay Description:Inhibition of mouse CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Mus musculus)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609674(CHEMBL5283284)
Affinity DataIC50:  26nMAssay Description:Inhibition of mouse CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609674(CHEMBL5283284)
Affinity DataIC50:  32nMAssay Description:Inhibition of human CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609670(CHEMBL5277468)
Affinity DataIC50:  42nMAssay Description:Inhibition of human CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Mus musculus)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609670(CHEMBL5277468)
Affinity DataIC50:  53nMAssay Description:Inhibition of mouse CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609644(CHEMBL5288271)
Affinity DataIC50:  180nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609662(CHEMBL5275093)
Affinity DataIC50:  210nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609647(CHEMBL5291055)
Affinity DataIC50:  250nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609664(CHEMBL5270156)
Affinity DataIC50:  420nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609665(CHEMBL5288933)
Affinity DataIC50:  430nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Mus musculus)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609669(CHEMBL5288393)
Affinity DataIC50:  440nMAssay Description:Inhibition of mouse CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609668(CHEMBL5287919)
Affinity DataIC50:  440nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609663(CHEMBL5288354)
Affinity DataIC50:  440nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609652(CHEMBL5284514)
Affinity DataIC50:  570nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609669(CHEMBL5288393)
Affinity DataIC50:  580nMAssay Description:Inhibition of human CTPS1 preincubated for 10 mins followed by substrate addition and measured after 30 to 60 mins by RFMS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609661(CHEMBL5278356)
Affinity DataIC50:  950nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609643(CHEMBL5266038)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609666(CHEMBL5280120)
Affinity DataIC50:  4.47E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609660(CHEMBL5270880)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609667(CHEMBL5279706)
Affinity DataIC50:  7.18E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609675(CHEMBL5288448)
Affinity DataIC50:  7.82E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609645(CHEMBL5270761)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609650(CHEMBL5279495)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609646(CHEMBL5270292)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609676(CHEMBL5279558)
Affinity DataIC50:  2.59E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609657(CHEMBL5283422)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609673(CHEMBL5267968)
Affinity DataIC50: <5.00E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609674(CHEMBL5283284)
Affinity DataIC50: <5.00E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609672(CHEMBL5287389)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609670(CHEMBL5277468)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609648(CHEMBL5279838)
Affinity DataIC50:  7.32E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609671(CHEMBL5280009)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609649(CHEMBL5269282)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609655(CHEMBL5272495)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609654(CHEMBL5291374)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609653(CHEMBL5271211)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609656(CHEMBL5286545)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609651(CHEMBL5287652)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609659(CHEMBL5285830)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609658(CHEMBL5270312)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCTP synthase 1(Homo sapiens)
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50609669(CHEMBL5288393)
Affinity DataIC50:  3.83E+5nMAssay Description:Inhibition of C-terminal FLAG-His8-tagged full length human CTPS1 preincubated for 10 mins followed by substrate addition by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed