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Report error Found 30 Enz. Inhib. hit(s) with Target = 'Calcium-activated potassium channel subunit beta'
LigandPNGBDBM86244(A-312110)
Affinity DataKi:  4.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86250(CAS_60559-98-0 | NSC_43345 | P1075)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86250(CAS_60559-98-0 | NSC_43345 | P1075)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86247(BAY X 9228 | CAS_3038059 | NSC_3038059)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM86250(CAS_60559-98-0 | NSC_43345 | P1075)
Affinity DataKi:  20.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86247(BAY X 9228 | CAS_3038059 | NSC_3038059)
Affinity DataKi:  41.3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM86245(CAS_85371-64-8 | NSC_4826 | PINACIDIL)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86251(CAS_94535-50-9 | CROMAKALIM (-) | NSC_93504)
Affinity DataKi:  157nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86245(CAS_85371-64-8 | NSC_4826 | PINACIDIL)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86249(ZD 6169 | ZD-6169)
Affinity DataKi:  451nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86251(CAS_94535-50-9 | CROMAKALIM (-) | NSC_93504)
Affinity DataKi:  542nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86249(ZD 6169 | ZD-6169)
Affinity DataKi:  630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86246(zm244085)
Affinity DataKi:  671nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-1(Human)
Sanofi-Synthelabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50171290(5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86246(zm244085)
Affinity DataKi:  2.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-1(Human)
Sanofi-Synthelabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514444(CHEMBL4516172)
Affinity DataIC50:  602nMAssay Description:Inhibition of human BK alpha/beta4 channel expressed in HEK293T cells assessed as inhibition of K+ outward current fraction at -80 mV holding potenti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-1(Human)
Sanofi-Synthelabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50557680(CHEMBL4741793)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of BK (unknown origin) by patch clamp analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514444(CHEMBL4516172)
Affinity DataKd:  5.11E+5nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 (45 to 166 residues) incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514444(CHEMBL4516172)
Affinity DataKd:  9.75E+5nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 Q124A mutant incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514444(CHEMBL4516172)
Affinity DataKd:  7.82E+5nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 E104K mutant incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514445(CHEMBL4447233)
Affinity DataKd:  1.08E+8nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 (45 to 166 residues) incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514446(CHEMBL4524166)
Affinity DataKd:  5.50E+5nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 (45 to 166 residues) incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514447(CHEMBL4540900)
Affinity DataKd:  6.40E+5nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 (45 to 166 residues) incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit beta-4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514443(CHEMBL4563569)
Affinity DataKd:  1.10E+6nMAssay Description:Binding affinity to NT-495 fluorophore reagent labelled human BK beta4 (45 to 166 residues) incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed