Compile Data Set for Download or QSAR
Report error Found 24769 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor'
TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKd:  0.0930nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395582(CHEMBL2165133 | UNC10000004 | US9156822, 25)
Affinity DataEC50:  12nMMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395581(CHEMBL2165134 | UNC10000010 | US9156822, 28)
Affinity DataEC50:  18nMMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395583(CHEMBL2165132 | UNC10099973 | US9156822, 31)
Affinity DataEC50:  16nMMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185693(UNC10099988 | US9156822, 34)
Affinity DataEC50:  36nMMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185677(UNC10000003 | US9156822, 1)
Affinity DataEC50:  6.10nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataEC50:  126nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395569(CHEMBL2165119 | UNC10099975 | US9156822, 3 or UNC9...)
Affinity DataEC50:  13nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395570(CHEMBL2165118 | UNC10099983 | US9156822, 5)
Affinity DataEC50:  5.60nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185678(UNC10099984 | US9156822, 6)
Affinity DataEC50:  9.87E+3nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395575(CHEMBL2165140 | UNC10099996 | US9156822, 8)
Affinity DataEC50:  348nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185679(UNC10107953 | US9156822, 9)
Affinity DataEC50:  163nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185680(UNC10107954 | US9156822, 10)
Affinity DataEC50:  306nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185681(UNC10107955 | US9156822, 11)
Affinity DataEC50:  222nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185684(UNC10107962 | US9156822, 14)
Affinity DataEC50:  27nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185685(UNC10107966 | US9156822, 15)
Affinity DataEC50:  13nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185687(UNC10107968 | US9156822, 17)
Affinity DataEC50:  0.200nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185688(UNC10107969 | US9156822, 18)
Affinity DataEC50:  0.100nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395572(CHEMBL2165116 | UNC10099976 | US9156822, 20)
Affinity DataEC50:  9.70nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395578(CHEMBL2165137 | UNC10099993 | US9156822, 21)
Affinity DataEC50:  21nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395576(CHEMBL2165139 | UNC10099995 | US9156822, 23)
Affinity DataEC50:  9.80nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395582(CHEMBL2165133 | UNC10000004 | US9156822, 25)
Affinity DataEC50:  3.70E+3nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185690(UNC10000007 | US9156822, 26)
Affinity DataEC50:  4.60E+4nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395585(CHEMBL2165129 | UNC10000009 | US9156822, 27)
Affinity DataEC50:  1.00E+3nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395581(CHEMBL2165134 | UNC10000010 | US9156822, 28)
Affinity DataEC50:  5.70nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395583(CHEMBL2165132 | UNC10099973 | US9156822, 31)
Affinity DataEC50:  5.70nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185693(UNC10099988 | US9156822, 34)
Affinity DataEC50:  512nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185694(UNC10107957 | US9156822, 37)
Affinity DataEC50:  11nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185695(UNC10108010 | US9156822, 38)
Affinity DataEC50:  1.80nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185697(UNC10108018 | US9156822, 41)
Affinity DataEC50:  0.400nMpH: 7.4Assay Description:HEK293T cells co-expressing the cAMP biosensor GloSensor-22F (Promega) and hD2 receptors were seeded (10,000 cells/20 ul/well) into white, clear-bott...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185677(UNC10000003 | US9156822, 1)
Affinity DataEC50:  3.10nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataEC50:  3.30nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395569(CHEMBL2165119 | UNC10099975 | US9156822, 3 or UNC9...)
Affinity DataEC50:  3.30nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395568(CHEMBL2165120 | UNC10099978 | US9156822, 4)
Affinity DataEC50:  2.80nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395570(CHEMBL2165118 | UNC10099983 | US9156822, 5)
Affinity DataEC50:  8nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185678(UNC10099984 | US9156822, 6)
Affinity DataEC50:  6.20nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395574(CHEMBL2165114 | UNC10099992 | US9156822, 7)
Affinity DataEC50:  23nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395575(CHEMBL2165140 | UNC10099996 | US9156822, 8)
Affinity DataEC50:  63nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185679(UNC10107953 | US9156822, 9)
Affinity DataEC50:  4.60nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185680(UNC10107954 | US9156822, 10)
Affinity DataEC50:  2.5nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185681(UNC10107955 | US9156822, 11)
Affinity DataEC50:  6.10nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185682(UNC10107958 | US9156822, 12)
Affinity DataEC50:  4.30nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185683(UNC10107959 | US9156822, 13)
Affinity DataEC50:  4nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185684(UNC10107962 | US9156822, 14)
Affinity DataEC50:  4.80nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185685(UNC10107966 | US9156822, 15)
Affinity DataEC50:  2.20nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185686(UNC10107967 | US9156822, 16)
Affinity DataEC50:  4.20nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185687(UNC10107968 | US9156822, 17)
Affinity DataEC50:  4.60nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185688(UNC10107969 | US9156822, 18)
Affinity DataEC50:  4.20nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM185689(UNC10108005 | US9156822, 19)
Affinity DataEC50:  8.5nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetD(2) dopamine receptor(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM50395572(CHEMBL2165116 | UNC10099976 | US9156822, 20)
Affinity DataEC50:  59nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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