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Report error Found 119 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase UHRF1'
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  1.93E+4nMAssay Description:Binding affinity to UHRF1 TTD (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity to UHRF1 Y188A/Y191A double mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  2.07E+4nMAssay Description:Binding affinity to UHRF1 TTD variant loop (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd: >1.11E+5nMAssay Description:Binding affinity to UHRF1 M224A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd: >1.83E+5nMAssay Description:Binding affinity to UHRF1 F278A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  4.50E+4nMAssay Description:Inhibition of His tagged UHRF1 tandem Tudor domain (unknown origin) using biotinylated-H3K9me3 peptide as substrate incubated for 1 hr by TR-FRET ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  2.90E+4nMAssay Description:Inhibition of His tagged UHRF1 tandem Tudor domain (unknown origin) using biotinylated-H3K9me3 peptide as substrate incubated for 1 hr by TR-FRET ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  2.92E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  4.51E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  5.67E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440605(CHEMBL2424677)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440606(CHEMBL2426376)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440607(CHEMBL2426375)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440608(CHEMBL2426374)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440609(CHEMBL2426373)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440610(CHEMBL2426368)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440611(CHEMBL2426367)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440612(CHEMBL2426366)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440613(CHEMBL2426365)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440614(CHEMBL2426364)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440560(CHEMBL2426363)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440561(CHEMBL2426362)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440562(CHEMBL2426361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440563(CHEMBL2426360)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440564(CHEMBL2426359)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440565(CHEMBL2426358)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440566(CHEMBL2426478)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440567(CHEMBL2426477)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440568(CHEMBL2426476)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440569(CHEMBL2424678)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440570(CHEMBL2426475)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440571(CHEMBL2426474)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440572(CHEMBL2426473)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440573(CHEMBL2426472)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440574(CHEMBL2426471)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440575(CHEMBL2426470)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440576(CHEMBL2426469)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440577(CHEMBL2426468)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440578(CHEMBL2426467)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440579(CHEMBL2426466)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440580(CHEMBL2426465)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440581(CHEMBL2426464)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440582(CHEMBL2426463)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440583(CHEMBL2426462)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440584(CHEMBL2426461)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440585(CHEMBL2426496)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440586(CHEMBL2426495)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440587(CHEMBL2426494)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50440588(CHEMBL2426493)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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